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2-(phenoxymethyl)-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}-1,3-oxazole-4-carboxamide
2-[methyl(2-phenylethyl)amino]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
2-(4-{5-amino-4-cyano-1,6-diazatricyclo[6.2.2.02,7]dodeca-2(7),3,5-trien-3-yl}phenoxy)propanoic acid
1-(5-{[2-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carbonyl)azocane
4-[(4-cyclohexyl-1,4-diazepan-1-yl)methyl]phenol
7-(1,3-benzothiazol-2-yl)-4-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1-benzylpiperidin-4-yl)-N-[(1r,4r)-4-hydroxycyclohexyl]piperidine-3-carboxamide
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
methyl (2S,4S)-4-[3-(3-fluorophenyl)benzamido]-1-[(3-hydroxyphenyl)methyl]pyrrolidine-2-carboxylate
1-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylic acid
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]acetamide
4-{[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-N-methylbenzene-1-sulfonamide
N,N-dimethyl-3-[1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidin-3-yl]propanamide
N-ethyl-3-(2-methylpropyl)-N-(oxan-4-ylmethyl)-1,2-oxazole-5-carboxamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(piperidin-1-ylmethyl)benzamide
methyl N-[4-(4,5-difluoro-2-hydroxyphenyl)phenyl]carbamate
(5S,9aS,9bS)-2-methyl-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-{4-[2-amino-6-(cyclopropylamino)pyrimidin-4-yl]piperazin-1-yl}pyridine-3-carboxamide
2-(5-cyclopropyl-1,2-oxazol-3-yl)-7-(4-fluorophenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-ethyl-4-(2-fluoro-6-methoxyphenyl)phenyl]acetamide
1-[(2-chlorophenyl)methyl]-3-(1-ethyl-1H-1,2,4-triazol-3-yl)-1-methylurea
5-{1-[(3-chloro-4-hydroxyphenyl)methyl]piperidin-4-yl}-5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)imidazolidine-2,4-dione
1-(4-{2-[(1R,5S)-6-azabicyclo[3.2.1]octane-6-carbonyl]-4-methoxyphenoxy}piperidin-1-yl)ethan-1-one
(2R)-2-amino-1-[2-(1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-phenylethan-1-one
1-[(4-fluorophenyl)methyl]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-{1-[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-4-yl}-2-methylpropan-1-ol
5-(2-ethoxyethyl)-3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
methyl 4-{[4-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]methyl}thiophene-2-carboxylate
N2-benzyl-6-(thiophen-2-yl)-1,3,5-triazine-2,4-diamine
1-(2-methoxyphenyl)-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperazin-2-one
N-[(8-{[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]acetamide
[(4aS,8aR)-6-butyl-1-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
6-(aminomethyl)-2-methyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
4-({[cyclopropyl(4-methoxyphenyl)methyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
(3S,4S)-1-(2-amino-4-methyl-1,3-thiazole-5-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
1-[(2R)-oxolan-2-ylmethyl]-5,5-diphenylpiperidin-2-one
1-methyl-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1H-indole
1-butyl-4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(2R,3R,6R)-5-(butane-1-sulfonyl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(propan-2-yl)-4-({3-[2-(pyridin-4-yl)pyridin-4-yl]pyrrolidin-1-yl}methyl)pyrimidine
2-(piperidin-1-yl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-2,3-dihydro-1H-indene-2-carboxamide
(3S,4S)-1-[(3-methoxyphenyl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1,9-dimethyl-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]-N-(2-hydroxy-3-methoxypropyl)benzamide
2-methyl-6-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2,3-dihydropyridazin-3-one
3-(4-chloro-1H-pyrazol-1-yl)-1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}propan-1-one
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-[4-(trifluoromethyl)benzoyl]piperidine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
{4-[(2-chlorophenyl)methyl]-1-(quinolin-2-ylmethyl)piperidin-4-yl}methanol