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ethyl 4-(piperidin-3-yl)piperazine-1-carboxylate
3-[1-(3,4-dimethylbenzoyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
3-{[2-(furan-2-yl)-1H-imidazol-1-yl]methyl}-2-methoxy-4,6-dimethylpyridine
1-(5-chloro-2-fluorobenzoyl)-3-(2-methoxyethyl)piperidine-3-carboxylic acid
N-(2-phenylethyl)-N-(propan-2-yl)pyridine-4-carboxamide
N-[(2-chlorophenyl)methyl]-3-[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]propanamide
(2S,4R)-4-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetamido]-N-ethyl-1-(oxan-4-yl)pyrrolidine-2-carboxamide
1-benzyl-5-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[3-(propan-2-yloxy)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
2-{4-[(4-ethynylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
1-(2-methoxyphenyl)-4-[2-(1H-pyrazol-1-ylmethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
1-{4-[4-(pyridin-4-yl)piperidine-1-carbonyl]phenyl}imidazolidine-2,4-dione
1-[(2,3-dimethoxyphenyl)methyl]-3-[(4,4-dimethylpiperidin-1-yl)methyl]-3-hydroxypiperidin-2-one
4-(2-methoxy-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)-1-methylpiperidine
{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-8-methylquinolin-3-yl}methanol
4-[2-(2-methoxy-4-methylphenoxymethyl)-1,3-oxazole-4-carbonyl]thiomorpholine
N-[(5-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-{[1-(4-acetylpiperazin-1-yl)hex-5-en-2-yl]oxy}-2-methoxypyridine-3-carbonitrile
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-1-ylmethyl)piperidin-3-yl]-N-[(3,4,5-trimethoxyphenyl)methyl]propanamide
3-benzyl-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
1-(1,2-oxazol-5-ylmethyl)-3-[5-(3-oxo-3-phenylpropyl)-1,3,4-thiadiazol-2-yl]urea
4-(2,1,3-benzothiadiazol-4-yl)-3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-methoxy-4-oxo-N-[2-(piperidin-1-yl)ethyl]-1,4-dihydropyridine-2-carboxamide
5-[4-(1H-pyrazol-1-ylmethyl)piperidine-1-carbonyl]-N-[2-(pyridin-4-yl)ethyl]pyridin-2-amine
2-[2-(4-chloro-1H-pyrazol-1-yl)acetyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
3-(3-chlorobenzoyl)-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
6-{[3-(methylsulfanyl)propyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
2-{4-[(3,5-dimethylphenyl)methyl]-1-(2,2-dimethylpropyl)piperazin-2-yl}ethan-1-ol
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-[3-(propan-2-yloxy)benzoyl]piperidine
(3aS,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-[3-(trifluoromethyl)pyridin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
ethyl 4-{2-[3-(2-methoxyphenyl)-1-(3-methoxypropyl)-2,5-dioxopyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)-2-(3,4,5-trimethoxyphenyl)ethan-1-one
1-cyclohexyl-3-(2-methyl-1,3-benzothiazol-5-yl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]urea
methyl 5-{3-[(naphthalen-1-ylformamido)methyl]piperidin-1-yl}-5-oxopentanoate
3-{5-[(trimethyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
[(3-chloro-5-fluoro-4-methoxyphenyl)methyl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amine
4-{6-amino-4-[2-(carboxymethoxy)phenyl]-5-cyanopyridin-2-yl}benzoic acid
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[(2-methylphenyl)methyl]pyrimidine-5-carboxamide
3-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-{[(6-ethoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl](methyl)amino}-N-methylbutanamide
3-[(2-oxoazonan-1-yl)methyl]benzonitrile
3-({2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)benzonitrile
(3R,5S)-N-butyl-5-(morpholin-4-ylmethyl)piperidine-3-carboxamide
1-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetyl}-N-(1-methoxypropan-2-yl)piperidine-4-carboxamide
N-[3-(1,3-benzoxazol-2-yl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
6-chloro-8-methyl-3-[1-(pyridin-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
3-(2-methyl-1H-imidazol-1-yl)-N-[1-methyl-4-(propan-2-yloxy)-1H-indazol-3-yl]propanamide
N1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}pentane-1,5-diamine