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3-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-indole
benzyl 3-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]pyrrolidine-1-carboxylate
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
methyl 3-(furan-3-ylmethyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
2-{3-cyclopropyl-5-[(1S)-2-methyl-1-(methylamino)propyl]-1H-1,2,4-triazol-1-yl}acetic acid
N-[3-(1H-imidazol-1-yl)propyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
2-{1-[1-(propan-2-yl)piperidin-4-yl]-4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
2-{5-[6-amino-5-cyano-4-(2-methoxypyrimidin-5-yl)pyridin-2-yl]thiophen-3-yl}acetic acid
7-chloro-3,5-dimethyl-N-(oxan-4-yl)-1-benzofuran-2-carboxamide
3-(3-methoxyphenyl)-N-propyl-N-(pyridin-3-ylmethyl)propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-3-yl}piperazine
2-(2,5-dimethylfuran-3-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3,4-dimethylphenoxy)ethan-1-one
N-{3-[3-(hydroxymethyl)-8-methylquinolin-2-yl]phenyl}acetamide
6-(2-aminoethyl)-2-(3-{[propyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(2,5-dioxoimidazolidin-4-yl)propanamide
2-methoxy-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-5-sulfamoylbenzamide
ethyl 4-({[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl](methyl)amino}methyl)-1H-pyrazole-3-carboxylate
(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
4-(4-methylphenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
N-(propan-2-yl)-2-{4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidin-4-amine
3-({1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidin-3-yl}methyl)benzamide
N-[(2R,3R)-1'-[(1-ethyl-1H-imidazol-2-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
N,N-diethyl-1-{[4-(1H-pyrazol-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidine-3-carboxamide
2-amino-4-{[(2-methoxyphenyl)methyl]amino}quinazoline-6-carboxylic acid
5-(2-fluorophenyl)-N-methyl-N-[2-(morpholin-4-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-(quinazolin-4-yloxy)ethan-1-one
(5S,9aS,9bS)-5-(1-benzofuran-2-yl)-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}-1,4-oxazepan-6-yl)methanol
6-(dimethylamino)-N-methyl-N-[1-(pyridin-3-yl)pentyl]pyridine-3-carboxamide
N-[1-(1-cyclobutylpiperidin-4-yl)-2-(2-fluorophenyl)ethyl]-N-methylthiophene-2-carboxamide
1-(2-methylphenyl)-4-(2-propoxybenzoyl)piperazin-2-one
4-(1,7-dimethyl-1H-indole-2-carbonyl)-3-methyl-1-phenylpiperazin-2-one
N-cyclopropyl-1-{2-[1-(3-phenylpropanoyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
(4aR,7aS)-1-methyl-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(1H-imidazol-1-yl)propyl]-2-[4-(methylsulfanyl)phenyl]-1H-imidazole
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)-1,3-oxazole-5-carboxamide
3-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1-[2-(oxan-2-yl)ethyl]urea
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
5-[5-(methoxymethyl)furan-2-carbonyl]-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]quinoline
N-[4-(3-fluorophenyl)phenyl]-1-(furan-3-carbonyl)piperidine-3-carboxamide
{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(oxan-4-yl)ethyl]amine
1-(adamantan-2-yl)-4-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
(2S,4R)-1-(cyclobutylmethyl)-N-(propan-2-yl)-4-[2-(pyridin-4-yl)acetamido]pyrrolidine-2-carboxamide
3,4,7-trimethyl-2-[2-(trifluoromethyl)morpholine-4-carbonyl]-1H-indole
3-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-5-(trifluoromethyl)-1H-1,2,4-triazole
9-(2-phenoxyethyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one