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methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl})[1-(thiophen-2-yl)ethyl]amine
2-phenoxy-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}[(2-fluoro-4,5-dimethoxyphenyl)methyl]methylamine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[1-(2-methoxyethyl)piperidin-3-yl]methyl})amine
2-ethyl-7-[(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)methyl]-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-5-one
3-{imidazo[1,2-a]pyridin-2-yl}-N-[1-(thiophen-3-yl)propan-2-yl]propanamide
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-2-(2-phenylethyl)piperidine
(2S,4S)-1-[(4-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N,N-dimethyl-N'-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)butanediamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-methyl-1H-indole-6-carboxamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
3-benzyl-8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)oxolane-2-carboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[3-(2-methyl-1H-imidazol-1-yl)propyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
6-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)piperidin-4-yl]pyrrolidin-2-one
3-(3-fluorophenyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
4-(2-fluorophenoxy)-1-[2-(pyridin-3-yl)acetyl]piperidine-4-carboxylic acid
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl][(2,2-dimethyloxan-4-yl)methyl]methylamine
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}({[2-fluoro-5-(trifluoromethyl)phenyl]methyl})amine
1-methyl-N-[(6-methylquinolin-5-yl)methyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
3-[(3R,4S)-4-(dimethylamino)-1-[(furan-2-ylmethyl)carbamoyl]piperidin-3-yl]propanoic acid
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2,3-dihydro-1H-inden-1-yl)-N-methylacetamide
5-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
N-[(3R,4S)-1-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
4-{3-[(4-methoxyphenyl)amino]piperidine-1-carbonyl}-N,N-dimethylpiperidine-1-carboxamide
1-methyl-4-{3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}piperidin-4-ol
N-ethyl-4-methanesulfonyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
methyl 3-(2,4-dimethylbenzamido)-6-{[(furan-2-ylmethyl)(methyl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
(3S,4R)-1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
1-[1-(pyridin-2-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
N-(oxolan-2-ylmethyl)-3-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)propanamide
(1R,2S)-N1-butyl-N2-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]cyclohexane-1,2-dicarboxamide
N-[4-(3-fluorophenyl)phenyl]-1-(4-oxopentanoyl)piperidine-3-carboxamide
1-(4-methoxyphenyl)-5-methyl-4-[3-(thiophen-2-yl)propanoyl]piperazin-2-one
N-{2-[3-phenyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
N-[(1-ethyl-5-oxopyrrolidin-3-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-{[1-(azepane-4-carbonyl)piperidin-4-yl]methyl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-fluorophenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1H-pyrazole-4-carboxamide
5-(2-cyclopentylacetamido)-N-[(2,3-difluorophenyl)methyl]-1-methyl-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamide
3-(3-aminopyrrolidine-1-carbonyl)-N-[2-(pyridin-3-yl)ethyl]benzene-1-sulfonamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
8-{[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-[4-(4-{[(6-methylpyridin-2-yl)methyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
1-[9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
5-oxo-1-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidine-3-carboxylic acid