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1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-diethylpyrrolidin-3-amine
(1R,5S,8S)-3-[(6-chloroquinolin-2-yl)methyl]-N,N-dimethyl-3-azabicyclo[3.2.1]octan-8-amine
3-hydroxy-3-{[(3-hydroxy-3-methylbutyl)(methyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(1R,3S,5S)-8-[2-amino-6-(diethylamino)pyrimidin-4-yl]-8-azabicyclo[3.2.1]octan-3-ol
7-[1-(2-hydroxyethyl)-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]-3-methyl-3,4-dihydroquinazolin-4-one
1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(3-methoxybenzoyl)piperazine
5,6-dimethyl-2-(2-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}-2-oxoethyl)-2,3-dihydropyridazin-3-one
methyl 2-(2-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylformamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
2-acetyl-8-{[4-(propan-2-yl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
ethyl 1-(pyridine-4-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-(1H-indol-1-ylmethyl)-N-methyl-N-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazole-3-carboxamide
2-(4-methoxyphenyl)-7-methyl-3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}quinoline
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-{3-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-oxopropyl}-N-methylmethanesulfonamide
1-[(2E)-2-methylbut-2-en-1-yl]-4-(2-phenoxyethyl)-1,4-diazepan-5-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-amine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}propan-1-one
N-(1-{1-[3-(1H-pyrazol-1-yl)propyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
3-{2-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-{[(1R,3S,5S)-3-hydroxy-8-azabicyclo[3.2.1]octan-8-yl]methyl}-N-(1H-indazol-5-yl)benzamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-4-phenylbutanamide
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-phenylpropyl)acetamide
N-(4-chlorophenyl)-3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
methyl 3-(2-methoxyacetamido)-1-methyl-5-({[3-(2-methylphenyl)phenyl]methyl}amino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[4-(3-methoxyphenyl)-1H-imidazol-2-yl]pyrrolidin-2-one
2-{2,5-dioxo-3-phenyl-1-[2-(pyridin-2-yl)ethyl]pyrrolidin-3-yl}-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
8-(6-cyclopropylpyrimidin-4-yl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-ethoxyethyl)-2-oxo-N-[2-(3-oxopiperazin-1-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
6-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]pyridine-2-carboxylic acid
[2-({4-[(6-methoxypyridin-3-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
N-[2-(2,5-dioxopyrrolidin-1-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
2-[1-(cyclohexylmethyl)-4-[(2,4-difluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1-methanesulfonylpyrrolidine-2-carboxamide
5-(3,4-dimethylphenoxymethyl)-N-[(2-methoxyphenyl)methyl]-1,2-oxazole-3-carboxamide
5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
(1R,5S)-3-[1-(methoxymethyl)cyclobutanecarbonyl]-3,8-diazabicyclo[3.2.1]octane
1-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]-1,2,3,4-tetrahydronaphthalene-1-carboxylic acid
2-{4-[3-(2,5-dihydro-1H-pyrrole-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
3-(piperidine-1-carbonyl)-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine
4-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-6-ethylpyrimidine
N-cyclopropyl-4-(2,5-dihydro-1H-pyrrol-1-yl)-7-(1H-imidazol-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
N-[(3,4-difluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[(3-methylthiophen-2-yl)formamido]methyl}benzoate
4-({9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)benzonitrile
(3R,4R)-1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-3,4-dimethylpyrrolidin-3-ol
N-ethyl-2-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]propanamide
3-{[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]oxy}-N-cyclopropyl-4-methoxybenzamide
(3S,4R)-4-(2-methoxyphenyl)-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}pyrrolidine-3-carboxylic acid
6-(propan-2-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyridazin-3-amine
9-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-2-methyl-2,9-diazaspiro[5.5]undecan-3-one