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1-cyclohexyl-4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperazine
N-(3-methoxypropyl)-4-methyl-N-{[6-(2-methylphenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}benzamide
4-[(4-ethoxyphenyl)methyl]-3-[2-(morpholin-4-yl)-2-oxoethyl]piperazin-2-one
1-(4-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
4-(5-{1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-1,2,3-triazol-4-yl}pyrimidin-2-yl)morpholine
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-3-(3-hydroxyquinoxalin-2-yl)propanamide
6-(4-methoxypiperidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-(3-{3-cyclopentyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidin-1-yl)pyridine
3-{2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
5-(3,4-dimethylphenoxymethyl)-N-{[3-(methylsulfanyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
1-{[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}cyclopentane-1-carboxamide
5-[(dimethylsulfamoyl)amino]-N,1-dimethyl-2-(2-methylpropyl)-N-(oxan-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(3-fluoropyridin-4-yl)-4-(4-methoxyphenyl)-2-methylpiperazine
3-(1H-pyrazol-1-yl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(propane-2-sulfonyl)piperidine
N-[2-(furan-2-yl)ethyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]amino}pyrimidine-5-carboxylic acid
1-cyclohexanecarbonyl-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
4-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-5-phenyl-2-(pyridin-4-yl)pyrimidine
(1R,5R)-6-(2-methoxyethyl)-3-(2-methyl-4-phenylpyrimidine-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-chloro-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}pyridin-2-amine
N-methyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]-2,3-dihydro-1H-indene-1-carboxamide
N-[3-(4-fluorophenyl)phenyl]-1-(pent-4-enoyl)piperidine-3-carboxamide
1'-[(3-methyl-1,2-oxazol-5-yl)methyl]-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-(4-chlorophenyl)-4-{2-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]ethyl}piperazine
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-2-oxo-2-(pyridin-3-yl)acetamide
1-[1-(2-cyclopropyl-1,3-benzoxazole-6-carbonyl)piperidin-4-yl]-3-phenylpropan-1-ol
3-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-[4-(1H-imidazol-1-yl)phenyl]urea
4-[1-(oxolane-3-carbonyl)piperidin-4-yl]-5-phenyl-2-(pyridin-3-yl)pyrimidine
1-[(2-fluorophenyl)methyl]-4-(1H-pyrazole-4-carbonyl)piperazin-2-one
(1R,5S,6S)-6-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-3-azabicyclo[3.1.0]hexane
2-methyl-N-(1,2,2,6,6-pentamethylpiperidin-4-yl)-6-(piperidin-4-yl)pyrimidin-4-amine
4-{3-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
N,1-dimethyl-3-propyl-N-[1-(1,3-thiazol-5-yl)ethyl]-1H-pyrazole-5-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-(2H-indazol-2-yl)acetamide
2-amino-4-cyclopropyl-6-(3,5-difluorophenyl)pyridine-3-carbonitrile
(3R,5S)-N-[2-(dimethylamino)ethyl]-5-(3-fluorophenoxymethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-5-ethyl-1,3-oxazole-4-carboxamide
methyl 3-{[3-(morpholin-4-yl)piperidin-1-yl]sulfonyl}thiophene-2-carboxylate
(3S,4S)-1-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(propan-2-yloxy)pyrrolidin-3-ol
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[3-(2-hydroxyphenyl)propyl]benzamide
2-(4-methylphenoxy)-1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}ethan-1-one
2-(1H-indol-1-yl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-ethyl-5-{[2-(3-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidin-2-amine
2-(2,3-dihydro-1H-indol-1-yl)-2-oxo-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)acetamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-cycloheptylpiperidin-3-ol
2-{1-[(4-methoxypiperidin-1-yl)sulfonyl]pyrrolidin-3-yl}benzoic acid
1-ethyl-3-(propan-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-cyclopropyl-N-[(8-methoxyquinolin-5-yl)methyl]-N,4-dimethylpyrimidine-5-carboxamide