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2-acetamido-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
1-(4-fluorophenyl)-4-(thian-4-yl)-1,4-diazepane
1-({1-[6-(4-hydroxypiperidin-1-yl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-methoxy-6-[3-(1H-pyrazol-3-yl)phenyl]pyrimidine
1-{3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-fluoro-4-methoxyphenyl)-1-[3-methyl-1-(pyridin-3-yl)butyl]urea
(2S,4S)-1-[(2-chlorophenyl)methyl]-4-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
ethyl 4-(3-phenylpropyl)-1-(thiolan-3-yl)piperidine-4-carboxylate
({4-[1-(2,3-difluorobenzoyl)piperidin-2-yl]phenyl}methyl)dimethylamine
6-(2-hydroxyethyl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-(3-methoxyphenyl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N,5-dimethyl-4-[(2-phenylethyl)amino]-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
1-(4-{2-[2-(hydroxymethyl)piperidine-1-carbonyl]-4-methoxyphenoxy}piperidin-1-yl)ethan-1-one
1-(5-chlorothiophene-2-carbonyl)-4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine
1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
7-{4-[(butylsulfanyl)methyl]-5-methylfuran-2-carbonyl}-3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
2-hydroxy-2-(4-methoxyphenyl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
6-methyl-5-[5-(3-phenoxypropyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1H-imidazol-1-yl)-3-methylbutan-2-yl]benzamide
4-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-1-(2-methoxyphenyl)piperazin-2-one
5-methyl-4-(1-methyl-1H-pyrazol-5-yl)-2-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine
2-butyl-8-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
1-methyl-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1,5-dimethyl-N-{[5-methyl-7-(2-methylquinolin-6-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-3-carboxamide
2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(oxolan-2-ylmethyl)acetamide
1-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(1-methyl-1H-pyrrol-3-yl)ethan-1-one
N,1-dimethyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-{1-[4-(1H-imidazol-1-yl)butanoyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-({1-[(2E)-2-methylpent-2-en-1-yl]pyrrolidin-3-yl}methyl)-1,3-thiazole-5-carboxamide
4-ethyl-3-({1-[2-(2-ethylpiperidin-1-yl)acetyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[(2,4-dimethoxyphenyl)methyl]-1-(propan-2-yl)piperazin-2-yl}ethan-1-ol
N-[(3R,4S)-4-cyclopropyl-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]-2-(2-oxopyrrolidin-1-yl)acetamide
3-(2-methoxyethyl)-1-[2-(propan-2-yl)phenyl]-3-(1,3-thiazol-2-ylmethyl)urea
[(2-methyl-1H-imidazol-4-yl)methyl][(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
N-{[4-(cycloheptyloxy)-3-methoxyphenyl]methyl}-2-methyl-N-(pyridin-2-ylmethyl)propanamide
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-[(2-methyl-1,3-thiazol-4-yl)methyl]-decahydro-2,7-naphthyridine-2-carboxamide
1-methyl-4-(1-{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}ethyl)piperazine
5-methoxy-2-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}-1,4-dihydropyridin-4-one
N-methyl-2-(3-{3-[3-(pyrrolidin-1-ylmethyl)phenyl]phenyl}-1H-pyrazol-1-yl)acetamide
{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-2,5-dihydro-1H-pyrrol-2-yl}methanol
2-(3-methoxyphenyl)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperidine
2-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}-7-methyl-2,7-diazaspiro[4.4]nonane
(1S,5R)-6-propyl-3-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-methoxybutan-2-yl)-5-[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazole
N,N-dimethyl-2-[4-(3-methyl-1H-pyrazol-4-yl)phenyl]acetamide
(1S,2R)-N1-ethyl-N1-(2-hydroxyethyl)-N2-propylcyclohexane-1,2-dicarboxamide
2-[4-(furan-3-ylmethyl)morpholin-3-yl]-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]acetamide