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3-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-benzoxazole
ethyl 4-[2-(2,3-dihydro-1H-inden-1-yl)acetamido]piperidine-1-carboxylate
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-phenylethyl)morpholine
8-(3-{imidazo[1,2-a]pyridin-2-yl}propanoyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(methanesulfonylmethyl)-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}pyridine
N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-2-(furan-2-yl)pyrrolidine-1-carboxamide
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-[(3-methylpyridin-2-yl)methyl]acetamide
(1H-1,3-benzodiazol-2-ylmethyl)(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-methyl-4-[2-(propan-2-yl)pyrimidin-4-yl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-(2-chloro-5-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
5-{2-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
propan-2-yl 4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxylate
N-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
N-{[5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
{[7-chloro-4-(morpholin-4-yl)quinazolin-2-yl]methyl}[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]methylamine
3-chloro-N-(2-methoxyethyl)-4-[(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)oxy]benzamide
N-methyl-2-{[(2-propylphenyl)carbamoyl]amino}pentanamide
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
3-[(dimethylamino)methyl]-1-[(6-methylquinolin-5-yl)methyl]pyrrolidin-3-ol
(1R,5S)-6-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-6-azabicyclo[3.2.1]octane
5-tert-butyl-4-{[2-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}furan-2-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-(cyclopropylmethyl)-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
ethyl 5-benzyl-1-[2-(dimethylamino)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
7-cyclopentyl-2-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-(2,3-dihydro-1H-inden-2-yl)-2-[(3,4-dimethoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(1,2-oxazinan-2-yl)propanamide
2-(oxolane-3-carbonyl)-8-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
4-(piperidin-1-ylmethyl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
7-(2-methoxyphenyl)-2-(pyridin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-cyclopentyl-N-[(2,3-difluoro-4-methylphenyl)methyl]-6-oxopiperidine-3-carboxamide
N-ethyl-N-(3-phenylpropyl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2-{1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
4-[(2S)-1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}pyrrolidine-2-carbonyl]morpholine
6-[4-(3-methoxypropyl)piperazin-1-yl]-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-4-one
6-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
(1S,5R)-6-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-4-amino-N,N-diethyl-1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
2-(4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
1-[(diethylcarbamoyl)methyl]-N-{[4-(morpholin-4-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3S,9aR)-8-(3,5-difluorobenzoyl)-3-(1H-indol-3-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-benzyl-8-(2,2-diphenylethyl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)azepan-3-amine
1-methyl-N-(3-{5-methyl-4-[(thiophen-2-ylformamido)methyl]-1,3-oxazol-2-yl}phenyl)piperidine-3-carboxamide
1-ethyl-3-(propan-2-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
4-(3-fluorophenoxy)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)piperidine-4-carboxylic acid
N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-[(4-methylphenyl)methyl]acetamide
1-[(3-methylpyridin-2-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperazine