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6-[3-(4-phenoxybenzoyl)piperidin-1-yl]pyrimidin-4-amine
5-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}pyridine-2,4-diol
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-methoxyethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(morpholin-3-yl)acetamide
2-(5-{[5-(4-fluorophenyl)-2H-1,2,3,4-tetrazol-2-yl]methyl}-3-(2-methylpropyl)-1H-1,2,4-triazol-1-yl)pyridine
N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-5-methyl-1,2-oxazole-3-carboxamide
3-(4-fluorophenyl)-4-(1H-imidazol-2-ylmethyl)piperazin-2-one
1-(2-{[(cyclopropylmethyl)(methyl)amino]methyl}-6-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
7-[(3,4-difluorophenyl)methyl]-2-[3-(methylsulfanyl)propyl]-2,7-diazaspiro[4.5]decane
8-{2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carbonyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
3-[(pyridin-2-ylmethyl)sulfamoyl]-N-(pyrrolidin-3-yl)benzamide
N-ethyl-3-[({[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}(methyl)carbamoyl)amino]benzamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(pyridin-4-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[(1R,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-1H-1,3-benzodiazole
2-(1-benzyl-3-oxopiperazin-2-yl)-N-[3-(1H-pyrazol-1-yl)propyl]acetamide
3-{1-[(2-chloro-4-hydroxy-5-methoxyphenyl)methyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(4-cyanophenyl)-3-({[(1,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)benzamide
2-benzyl-N-(3-chloro-2,6-dimethylphenyl)-3-oxopiperazine-1-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
1-benzyl-2-(2-methoxyethanesulfonyl)-5-(pyrrolidin-1-ylmethyl)-1H-imidazole
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-(3-fluorobenzenesulfonyl)-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
1-[5-(3-chlorophenyl)-1,2,4-triazin-3-yl]-N,N-dimethylpyrrolidin-3-amine
4-(2-methylphenoxy)-1-(oxolan-3-ylmethyl)piperidine
6-[5-(1,4-dioxan-2-yl)-3-ethyl-1H-1,2,4-triazol-1-yl]-2-methyl-1,3-benzothiazole
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-1-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
1-cyclohexyl-6-(pyridin-2-ylmethoxy)-4-(quinoxalin-5-ylmethyl)-1,4-diazepan-2-one
4-{4-[(4-benzyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrrolidin-2-one
5-[(2-ethyl-1H-imidazol-1-yl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazole
3-[(3R,4S)-4-(dimethylamino)-1-[4-(propan-2-yl)benzenesulfonyl]piperidin-3-yl]propanoic acid
N-{2-cyclobutyl-7-[3-(dimethylamino)pyrrolidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-5-yl}-2-methoxyacetamide
1'-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-methyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-(butan-2-yl)-1-ethyl-3-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[4-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-[(2-amino-6-methylpyrimidin-4-yl)amino]-1-(2-phenylethyl)pyrrolidin-2-one
1-[2-(piperidin-2-yl)ethyl]-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-oxo-4-phenyl-N-[1-({[(4-phenyl-1,3-thiazol-5-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]butanamide
[(3R,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-3-yl]methanol
4-ethyl-N-{[3-(2-methoxyethoxy)phenyl]methyl}-5-methylpyrimidin-2-amine
1-[2-(morpholin-4-yl)ethyl]-5-(1,2-oxazinane-2-carbonyl)piperidin-2-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]piperazine
3-cyclopropyl-5-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-pyrazole
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N3-[2-(4-fluorophenyl)ethyl]-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
9-(cyclopropylmethyl)-1-methyl-4-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S)-2-amino-3-(1H-imidazol-4-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one