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1-cyclopentyl-N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methyl-6-oxopiperidine-3-carboxamide
9-{2-[3-(dimethylamino)pyrrolidin-1-yl]acetyl}-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]thian-4-amine
1-[(4-fluorophenyl)methyl]-2-oxo-3-(pyrimidin-2-ylmethyl)-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-ethyl-N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}piperidin-4-amine
7-(cyclopropylmethyl)-2-[(2,3-difluoro-6-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-methyl-8-[2-(2,2,2-trifluoro-1-phenylethoxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
5-benzyl-2-methyl-4-{1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl}pyrimidine
1-benzyl-8-(1-hydroxypropan-2-yl)-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[4-(benzyloxy)piperidin-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
N-[(3R,5S)-5-(methylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
N-{2-[methyl(phenyl)amino]propyl}-3-propyl-1H-pyrazole-5-carboxamide
N-[2-(3-methoxyphenyl)ethyl]-3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(3R,4S)-1-(carbamoylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-2-(2-methoxyethyl)piperidine
(2S,4R)-4-amino-1-[(1-benzyl-1H-indol-6-yl)methyl]-N-ethylpyrrolidine-2-carboxamide
1-[2-(1-butyl-3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-4-methylpiperazine
N-(2-methoxyethyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]-N-(propan-2-yl)acetamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(2,5-dioxoimidazolidin-4-yl)propanamide
[2-(tert-butylsulfanyl)ethyl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylimidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[3-(cyclohexyloxy)propyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
N-[(5-chloro-1H-indol-2-yl)methyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
(3S,4S)-1-{[2-(3-methylphenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperidine-3,4-diol
{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N,5-dimethyl-N-(1,3-thiazol-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
6-[3-(2-methylphenyl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
ethyl 3-[5-(5-acetylthiophen-3-yl)-4-phenyl-1H-imidazol-1-yl]propanoate
1-butyl-5-(1-cyclopropyl-1H-pyrrol-2-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1,4,6-trimethyl-3-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyridin-2-one
dimethyl(3-{2-[1-(5-methyl-1,3-oxazole-4-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
methyl (2S,4R)-1-[(2-chlorophenyl)methyl]-4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamido}pyrrolidine-2-carboxylate
1-(carbamoylmethyl)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidine-4-carboxamide
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[2-(thiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
3-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-8-methyl-1,4-dihydroquinolin-4-one
2-amino-4-(2-aminopyrimidin-5-yl)-6-(4-ethylphenyl)pyridine-3-carbonitrile
2-[benzyl({[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl})amino]ethan-1-ol
(1S,5R)-6-(cyclobutylmethyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
2,5-difluoro-N-(1-{7-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)benzamide
1-tert-butyl-N-(cyclohex-1-en-1-ylmethyl)-5-oxopyrrolidine-3-carboxamide
{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
(2S,4R)-4-amino-N-ethyl-1-(4,4,4-trifluorobutanoyl)pyrrolidine-2-carboxamide
3-{[3,3-bis(hydroxymethyl)piperidin-1-yl]methyl}-6-ethoxy-1,2-dihydroquinolin-2-one
8-cyclopropanecarbonyl-2-(4-methylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-2-oxoethyl)-4-(pyridin-3-ylmethyl)piperazin-2-one