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4-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
methyl 5-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-{1-[2-(methylamino)-1,3-thiazole-4-carbonyl]piperidin-3-yl}benzoic acid
N-benzyl-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-sulfonamide
4-(6-phenoxypyridin-3-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-(3-methyl-1H-pyrazol-1-yl)-N-{[4-(2-methylpropoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)propanamide
1-(pyridin-2-yl)-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
4-{5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]pyridin-2-yl}thiomorpholine
N-methyl-N-[(5-{[methyl(pyrazin-2-ylmethyl)amino]methyl}furan-2-yl)methyl]methanesulfonamide
1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-[(4-fluorophenyl)methyl]-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-(1H-indazol-5-yl)-5-oxopyrrolidine-3-carboxylic acid
N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]acetamide
2-(1-benzyl-4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
1-methyl-6-oxo-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,6-dihydropyridazine-3-carboxamide
6-[(3-fluorophenyl)methoxy]-4-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(2-methylpropyl)-1,4-diazepan-2-one
1-[(1-hydroxycyclohexyl)methyl]-5-methyl-5-phenylpiperidin-2-one
8-(3-fluoropyridin-4-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
(4aR,7aS)-1-(2-hydroxyethyl)-4-[(4-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-(5-methylpyrazine-2-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N,N-diethylpropanamide
(1S,5R)-6-(3-methyl-1,2-oxazole-5-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-fluoro-N-[(2-phenoxypyridin-3-yl)methyl]benzene-1-sulfonamide
2-[3-(2-chlorophenyl)-1-cyclopentyl-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[1-(1,2-oxazol-3-yl)ethyl]acetamide
6-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]pyrazine-2-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(1,2-oxazol-3-ylmethyl)acetamide
5-ethyl-2-{1-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-imidazol-2-yl}pyridine
N,4-dimethyl-4-[(3-methyl-1H-indol-2-yl)formamido]pentanamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-1,5-dimethyl-1H-pyrazole-3-carboxamide
4-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(pyridin-4-ylmethyl)piperidine-4-carboxamide
1-ethyl-4-{[4-(4-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]methyl}-1H-pyrrole-2-carbonitrile
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(3-methyl-1H-pyrazol-1-yl)acetamide
4-[2-methyl-2-(4-methylphenoxy)propanoyl]-1-(4-methylphenyl)piperazin-2-one
3-{benzyl[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amino}-1λ6-thiolane-1,1-dione
N-(1-hydroxy-3-methylbutan-2-yl)-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-{[3-(methylsulfanyl)phenyl]methyl}-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-(2-{[1-(2,3-dimethylphenyl)piperidin-4-yl]amino}ethyl)-N-methylmethanesulfonamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-phenoxyacetamide
1-{5-[3-(dimethylamino)phenyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazol-1-yl}butan-2-ol
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-{2-[4-(2-methoxyethyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
5-{[(1S,2R)-2-aminocyclobutyl]carbamoyl}-2,4-dimethyl-1H-pyrrole-3-carboxylic acid
4-(4-chlorophenoxy)-N-[1-(furan-2-yl)ethyl]piperidine-4-carboxamide
(3S,4S)-1-({3-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-4-(piperidin-1-yl)pyrrolidin-3-ol
ethyl 4-[1-(cyclohexylmethyl)-5-(ethylcarbamoyl)-4-oxo-1,4-dihydropyridine-3-carbonyl]piperazine-1-carboxylate
N-{2-[4-(dimethylamino)phenyl]ethyl}-4-(1H-pyrazol-4-yl)butanamide
3-(dimethyl-1,2-oxazol-4-yl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)propanamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
4-phenyl-N-{[1-(1,3-thiazol-2-ylmethyl)piperidin-3-yl]methyl}benzamide
7-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecan-4-yl]-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine