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2-[(4-chlorophenyl)methyl]-N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]benzamide
4-(2,3-dihydro-1H-inden-2-yl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)-1,4-diazepane-1-carboxamide
4-(2-oxo-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[(1S,2R)-2-(cyclohexylamino)cyclobutyl]-2-(4-methylphenoxy)ethane-1-sulfonamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-[(4-methyl-1,3-thiazol-5-yl)methyl]piperidine
3-{2-oxo-2-[2-(pyridin-2-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(6-hydroxypyrimidin-4-yl)methyl]amino}methyl)piperidin-2-one
5-(3-methylfuran-2-carbonyl)-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
7-(cyclohexylmethyl)-2-(5-propyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
[(3R,4S)-1-[(3-chloro-4-fluorophenyl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[(3S,7S,8aS)-3-(1H-indol-3-ylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-chloro-2-methylphenyl)urea
1-[2-methoxy-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
2-(adamantan-1-yl)-5-[(2S)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]pyrimidin-4-ol
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-(propan-2-yloxy)pyridazine
2-[1-(2,2-dimethylpropyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl]ethan-1-ol
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}azocane
4-(benzyloxy)-1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
(3S,4R)-4-(hydroxymethyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-ol
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
(4aR,7aS)-1-butanoyl-4-(5-ethylthiophene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(4-fluorophenyl)phenyl]-1-(pyridine-4-carbonyl)pyrrolidine-2-carboxamide
4-phenyl-1-(3-propyl-1H-pyrazole-5-carbonyl)azepane
1-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(1S,5R)-3-benzyl-6-[(4-fluoro-2-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
4-cyclohexyl-3-({4-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)-4H-1,2,4-triazole
ethyl 2-[(1R,5S,6S)-6-[4-(pyrimidin-2-yl)piperazine-1-carbonyl]-3-azabicyclo[3.1.0]hexan-3-yl]acetate
1-(3,5-dimethylphenyl)-4-{3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanoyl}piperazin-2-one
4-(1-benzothiophene-2-carbonyl)-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
[(1-cyclohexylpiperidin-3-yl)methyl](propyl)(pyridin-3-ylmethyl)amine
3-(azocan-1-yl)-N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]propanamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
ethyl 4-[1-(1H-indol-3-ylmethyl)piperidin-3-yl]piperazine-1-carboxylate
8-[1-(phenylamino)cyclopentanecarbonyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-5-oxopyrrolidine-2-carboxamide
2,6,8-trimethyl-N-(5-oxo-1-propylpyrrolidin-3-yl)quinoline-4-carboxamide
benzyl({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
1-[3-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)pyridin-2-yl]piperidin-3-ol
4-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1-cyclopentylpiperazin-2-one
N-(1-cycloheptylpiperidin-3-yl)-2,6-dimethoxybenzamide
3-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-1-(thiomorpholin-4-yl)propan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
1-(3-{4-[methyl(oxan-2-ylmethyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
2-(2-chloro-4-fluorophenyl)-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
(4aS,8aR)-1-(3-aminopropyl)-6-[(3-methyl-1-benzofuran-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
4-[4-(piperidine-1-carbonyl)phenoxy]-1-(thiolan-3-yl)piperidine
2-(1H-indol-5-yl)pyridine-3-carbonitrile
1-(2-methylpropyl)-6-(pyridin-2-ylmethoxy)-4-[2-(pyridin-3-yl)quinoline-4-carbonyl]-1,4-diazepan-2-one
N-methyl-5-(naphthalen-2-yl)-N-(oxan-4-ylmethyl)-1,2,4-triazin-3-amine
N-{2-[7-(2,3-dihydro-1-benzofuran-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-(4-fluorophenyl)acetamide
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide