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5-(2-methoxyacetamido)-1-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
N-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-6-methoxypyrimidin-4-amine
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole-5-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[(3-hydroxyphenyl)methyl]-N-methylbutanamide
N-{4-[2-(1H-indazol-1-yl)acetamido]phenyl}-5-methylfuran-2-carboxamide
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,6-trifluorobenzamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3-methyl-1-benzofuran-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(2-oxopyrrolidin-1-yl)benzamide
N-methyl-2-{3-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}-N-(propan-2-yl)acetamide
1-(4-benzylpiperidin-1-yl)-3-[1-(2-hydroxyethyl)piperidin-4-yl]propan-1-one
1-(2-{[2-(pyridin-2-yl)ethyl]amino}pyrimidin-4-yl)pyrrolidin-3-ol
1-[3-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-3-oxopropyl]piperidin-2-one
2-{4-[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-6-yl}pyridine
5-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(thiophen-3-ylmethyl)piperidine-4-carboxylic acid
3-[(4,4-dimethylpiperidin-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
4-{1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
N-(1-{4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]phenyl}ethyl)acetamide
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-3-(1H-pyrazol-5-yl)piperidine
6-methoxy-N-[2-methyl-1-(pyridin-2-yl)propyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
4-[2-(2-fluoro-4-methylphenyl)pyridine-4-carbonyl]morpholine
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-5-propyl-1,2-oxazole-4-carboxamide
N-(3-{[(2,3-dihydroxypropyl)carbamoyl]amino}-2-methylphenyl)-2-methoxyacetamide
2-methyl-N-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-6-yl}-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
(2R,4S)-1-[2-(3-cyano-2-methyl-1H-indol-1-yl)acetyl]-4-hydroxypiperidine-2-carboxylic acid
3-{5-[2-(cycloheptylcarbamoyl)ethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-[(3,4-difluorophenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-(1-cyclopentyl-4-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
[(4-{2-[4-(2,5-dimethoxybenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(quinolin-6-ylmethyl)amine
2-{4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-(4-methyl-3-phenylpiperazin-1-yl)ethan-1-one
2-(methoxymethyl)-5-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}pyrimidine
3-fluoro-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
5-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-ethyl-9-(3-phenoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(4-{[3-(1H-imidazol-1-yl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-3-methylbut-2-en-1-one
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]acetamide
6-[(2-chloro-6-fluorophenyl)methyl]-N-[2-(2-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)(methyl)[1-(pyrimidin-4-yl)ethyl]amine
(4-benzyl-1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)methanol
N-[(2,4-difluorophenyl)methyl]-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-(2-{7-[(4-methoxy-2,3-dimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclohexanecarboxamide
5-(dimethyl-1,2-oxazole-4-carbonyl)-N-ethyl-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-({[2-(4-methoxyphenyl)-8-methylquinolin-3-yl]methyl}(methyl)amino)-N-methylacetamide
2-[({5-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(1H-1,2,4-triazol-1-yl)propanamide