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N-benzyl-4-oxo-1-(propan-2-yl)-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
5-methyl-1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-phenylpiperidin-2-one
1-{3-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N,N-dimethyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyridazin-3-amine
4-{[(2,5-dimethoxyphenyl)methyl]amino}-1-[(3-fluorophenyl)methyl]pyrrolidin-2-one
4-ethyl-1-methyl-3-{1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-methyl-4-(4-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}phenyl)butan-2-ol
3-{2-[4-(2-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
6-({[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
3-methyl-1-(2-methylpropyl)-4-(1,2-oxazole-3-carbonyl)piperazin-2-one
1'-(5-methyl-1,3-oxazole-4-carbonyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-({3-[2-(3-hydroxyphenyl)pyridin-4-yl]pyrrolidin-1-yl}methyl)-6-methylpyridin-3-ol
N-[2-(7-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]oxane-4-carboxamide
2-[2-(morpholin-4-ylmethyl)phenoxy]-5,6,7,8-tetrahydroquinoline-3-carbonitrile
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propane-1-sulfonyl)piperidine
5-[1-(furan-2-ylmethyl)pyrrolidin-2-yl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]thiophene-2-carboxamide
9-(6-aminopyridine-3-carbonyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(4-fluorophenyl)ethyl]-2-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]acetamide
2-[2-(3,5-difluoro-2-methoxyphenyl)phenoxy]propanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
5-({3-[(3-fluorophenyl)amino]piperidin-1-yl}methyl)-2-methoxyphenol
2-(2-amino-6-hydroxypyrimidin-4-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(3S)-3-({[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}amino)azepan-2-one
3-[(3R,4S)-4-(dimethylamino)-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]propanoic acid
methyl 6-{[bis(prop-2-en-1-yl)amino]methyl}-3-(thiophene-3-amido)thieno[2,3-b]pyridine-2-carboxylate
ethyl 4-[3-(3-hydroxyphenyl)-3-(4-hydroxyphenyl)propanoyl]piperazine-1-carboxylate
(1S,5R)-6-[(2-fluoro-5-methoxyphenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-[9-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
6-oxo-N-(2-phenoxyethyl)-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2-[1-(2-methylpropyl)-4-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]pyrimidine
7-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
2-ethoxy-5-({4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
ethyl 2-({10-azabicyclo[4.3.1]decane-10-carbonyl}amino)-1H-imidazole-5-carboxylate
2-[1-(2,2-dimethylpropyl)-4-(1H-indol-3-ylmethyl)piperazin-2-yl]ethan-1-ol
2-[9-(4-fluorobenzoyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
3-[2-(2,4-difluorophenyl)ethyl]-1-(furan-2-carbonyl)piperidine
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[2-(trifluoromethyl)benzoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]({[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl})methylamine
4-[1-(furan-3-carbonyl)piperidin-3-yl]-2-methyl-5-(3-methylphenyl)pyrimidine
2-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-ethoxyphenol
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
1-(6-methylpyridazin-3-yl)-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
[(3-{[1-(2,3-dimethyl-1H-indole-7-carbonyl)piperidin-4-yl]oxy}phenyl)methyl](furan-3-ylmethyl)methylamine
7-{[(3R,4R)-4-cyclobutyl-4-hydroxy-3-methylpiperidin-1-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-N,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidin-3-amine
{[2-(cyclopentyloxy)phenyl]methyl}(methyl)[1-(pyridin-4-yl)ethyl]amine