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7-chloro-4-methyl-2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
6-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[2-(pyrrolidin-1-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]ethan-1-one
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-[2-(methylsulfanyl)pyridine-3-carbonyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-{4-[2-hydroxy-4-(methylsulfanyl)butanoyl]-2-oxopiperazin-1-yl}benzonitrile
N-[(6-methylpyridin-2-yl)methyl]-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
3-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}pyrrolidin-3-ol
1-ethyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl](3-phenylpropyl)amine
2-(carbamoylamino)-N-[(5-ethylpyridin-2-yl)methyl]-N-methylacetamide
(4aR,7aS)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
(1r,4r)-4-{[4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-yl]amino}cyclohexan-1-ol
5-{[4-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]methyl}-1H-1,2,3,4-tetrazole
1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
5-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole
N-{3-[1-(cyclohex-2-en-1-yl)-1,2,3,6-tetrahydropyridin-4-yl]propyl}acetamide
methyl (2S)-2-{[6-(4-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-phenylpropanoate
1-{1-[(4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(piperidin-1-ylmethyl)piperidine
5-cyclopropyl-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,3,4-oxadiazol-2-amine
4-({[(3-methoxyphenyl)methyl](prop-2-en-1-yl)amino}methyl)-N-methylbenzene-1-sulfonamide
3-(1H-indol-5-yl)-4-methylbenzamide
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-4-(pyridin-3-yl)pyrimidin-2-amine
1-[3-(trimethyl-1H-pyrazol-4-yl)propanamido]cyclopentane-1-carboxamide
N-[2-(4-chlorophenyl)ethyl]-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
4-{[4-(dimethylamino)azepan-1-yl]methyl}-N-methylbenzene-1-sulfonamide
2-[(4-methoxyphenyl)methyl]-N-(3-methoxypropyl)-1,3-benzoxazole-6-carboxamide
N-benzyl-5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
methyl 3-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)propanoate
2-[5-(4-chloro-1-methyl-1H-indazol-3-yl)-4-phenyl-1H-imidazol-1-yl]ethan-1-ol
(1R,3R)-N1-[6-(morpholine-4-carbonyl)pyrazin-2-yl]cyclopentane-1,3-diamine
3-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(oxolan-2-ylmethyl)-N-propylpropanamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-(2-ethoxyphenyl)ethan-1-one
8-chloro-2-ethyl-4-(1H-pyrazol-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}acetamide
methyl({5-[(2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)[2-(oxan-2-yl)ethyl]amine
6-(2-chlorophenyl)-2-{3-[(4-methylpiperazin-1-yl)methyl]phenyl}-3,4-dihydropyrimidin-4-one
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-hydroxyethan-1-one
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N,N-dimethyl-3-[2-(morpholin-4-ylmethyl)phenoxy]pyrazin-2-amine
3-(3,4-dimethoxyphenyl)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
2-{3-cyclopropyl-5-[1-(pyridin-2-ylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
(2E)-1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-3-(1-methyl-1H-pyrazol-4-yl)prop-2-en-1-one
2-ethyl-N-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-2,5-dihydro-1H-pyrrole-1-carboxamide
2-(aminomethyl)-N-(2-chloro-5-methylphenyl)piperidine-1-carboxamide
N-(2-{6,8-dioxo-2,7-diazaspiro[4.4]nonan-2-yl}-2-oxoethyl)-N-(3-methylphenyl)methanesulfonamide
N-methyl-5-[methyl(2-methylpropyl)amino]-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
7-[(2-butyl-1H-imidazol-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-[7-(azocane-1-carbonyl)-1-ethyl-2-methyl-1H-1,3-benzodiazol-5-yl]benzenesulfonamide
3-{[ethyl(2-hydroxyethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide