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N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-(pyrazine-2-carbonyl)piperidin-4-amine
2-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-indole
3-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-methyl-1-benzofuran-5-carboxamide
4-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N,N,5-trimethylthieno[2,3-d]pyrimidine-6-carboxamide
4-{[4-(2-aminopropan-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-N-(3-fluorophenyl)piperidine-1-carboxamide
N-[(5-ethylpyridin-2-yl)methyl]-2-(4-fluorophenyl)-2-hydroxy-N-methylacetamide
N-(4-fluoro-3-methylphenyl)-3-{[(1H-imidazol-2-ylmethyl)(methyl)amino]methyl}benzamide
methyl({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-oxo-4-phenylbutanamide
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-ethyl-N-(2-hydroxyethyl)-5-(methoxymethyl)-1H-pyrazole-4-carboxamide
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-4-carboxamide
N-(1-benzylpiperidin-3-yl)-3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-{4-[(propan-2-yl)amino]piperidin-1-yl}benzamide
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(thiophene-3-carbonyl)pyrrolidin-3-amine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-4-methyl-N-(pyridin-3-ylmethyl)-1,2,3-thiadiazole-5-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
2-({[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}(methyl)amino)ethan-1-ol
2,6-dimethyl-3-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
4-[3-(1H-1,2,4-triazol-1-yl)propyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-(cyclopropylsulfamoyl)-5-(3,5-dimethoxyphenyl)benzoic acid
1-(cyclohexylmethyl)-6-oxo-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}piperidine-3-carboxamide
(3R,4R)-3-[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)(ethyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
(2R,6S)-2,6-dimethyl-N-[3-(methylsulfamoyl)phenyl]morpholine-4-carboxamide
N-{1-[5-(ethylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]ethyl}-1-phenylcyclohexane-1-carboxamide
1-(adamantan-1-yl)-4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazine
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-amine
methyl 3-{[1-(cyclopropylmethyl)-5-(2,3-difluorobenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]formamido}propanoate
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-9H-purin-6-amine
1-{5-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
2-methyl-6-{2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-2-oxoethyl}-6H,7H-[1,3]oxazolo[5,4-d]pyrimidin-7-one
N-[4-(2-fluorophenoxy)phenyl]-1-(2-methoxyacetyl)piperidine-4-carboxamide
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-methoxy-4-methyl-1,3-thiazole-5-carboxamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-benzyl-3-{[(butan-2-yl)amino]methyl}-N-methylpyridin-2-amine
8-(furan-3-ylmethyl)-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 4-(2-methoxyethyl)-1-(quinolin-4-ylmethyl)piperidine-4-carboxylate
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[2-(1H-imidazol-1-yl)ethyl]piperazine
9-methyl-3-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-3,9-diazaspiro[5.6]dodecane
3-(2,1,3-benzoxadiazol-5-ylmethyl)-8-fluoro-3,4-dihydroquinazolin-4-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-1-benzofuran-2-carboxamide
({4-[1-(2-ethylpyrimidine-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
1-methyl-N-[(1-methyl-1H-indol-2-yl)methyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
3-{[(1-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
3-({7-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-1,3-oxazolidin-2-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
2-(4-{4-[4-(4-methoxybenzoyl)piperazin-1-yl]piperidin-1-yl}phenyl)-1-(pyrrolidin-1-yl)ethan-1-one
5-chloro-2-(4-methoxy-2-methylphenyl)pyrimidine