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1-(2,2-dimethylpropyl)-4-[(6-methyl-2-phenylpyrimidin-4-yl)amino]pyrrolidin-2-one
N-[(5-{[(4-fluorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2,2-dimethyloxane-4-carboxamide
ethyl 1-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carbonyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
6-methyl-4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
5-methanesulfonyl-2-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]pyrimidin-4-amine
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-4-(morpholine-4-carbonyl)pyridin-2-amine
N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(N-methylmethanesulfonamido)propanamide
N-cyclopropyl-4-hydroxy-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-methylphenyl)pyrimidine-5-carboxamide
N-{2-[(3-methylpyridin-2-yl)amino]ethyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
6-ethyl-2-(1-ethyl-1H-pyrazol-4-yl)-4-(pyrrolidine-1-carbonyl)quinoline
6-(4-phenylbenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
2-(4-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-9-methoxy-7-oxo-3-(thiophene-3-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-(1,1-dioxo-1λ6-thian-4-yl)-N,5-dimethyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
N-{[3-(2-methoxyethoxy)phenyl]methyl}-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
7-(5-methyl-1H-indazole-3-carbonyl)-2,7-diazaspiro[4.5]decane
(3S,4S)-4-(dimethylamino)-1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidin-3-ol
4-[1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]morpholine
2-(3-hydroxypiperidin-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(3,4-dimethoxybenzoyl)-1-(thiophen-3-ylmethyl)piperidine
6-[4-(1H-indol-3-yl)butan-2-yl]-3-[(2-methoxyphenyl)methyl]-1-methyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-(trifluoromethyl)pyrimidin-2-amine
2-{1-[(3,4-difluorophenyl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
8-(2-methyl-4-phenylpyridine-3-carbonyl)-1-oxa-8-azaspiro[4.5]decane
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
1-{3-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]phenyl}ethan-1-one
5-(2-chlorophenyl)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]furan-2-carboxamide
N-(4-{[(1,2-oxazol-5-ylmethyl)carbamoyl]methyl}phenyl)butanamide
2-({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}(propan-2-yl)amino)ethan-1-ol
(3S,4R)-1-(1,4-dithiepan-6-yl)-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
1-(2-{[(6-methyl-2-propylpyrimidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
2-benzyl-9-(5-fluoro-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(4aR,8aS)-6-(4-fluorobenzoyl)-1-[4-(1H-imidazol-1-yl)benzoyl]-decahydro-1,6-naphthyridine
1,3-dimethyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-butyl-N-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-4-methyl-3-oxopiperazine-1-carboxamide
1-{4-[5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidin-4-yl]piperidin-1-yl}-4-(thiophen-2-yl)butan-1-one
N-[(4-chlorophenyl)methyl]-2-propanoyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)furan-2-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}cyclopropanecarboxamide
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-N-(4-oxo-4H-chromen-6-yl)piperidine-1-carboxamide
methyl({[2-(methylsulfanyl)pyrimidin-5-yl]methyl})[(1-phenylpyrrolidin-3-yl)methyl]amine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(pyridin-2-yl)-N-(pyridin-3-ylmethyl)propanamide
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-ethyl-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
N-(2-hydroxybutyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
4-(1H-imidazol-1-yl)-1-phenylmethanesulfonylpiperidine-4-carboxylic acid
N-(2-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}ethyl)acetamide
1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1,4-diazepan-5-one
3-(benzyloxy)-1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)piperidine
5-{5-[morpholin-4-yl(pyridin-3-yl)methyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole