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1-[(3R,4R)-3-{[ethyl(2-hydroxyethyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
9-(cyclopropylmethyl)-1-methyl-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methyl-6-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-amine
(3R)-1-[3-(3-hydroxy-3-methylbutyl)benzoyl]pyrrolidin-3-ol
3-[(4-methoxy-4-methylpentan-2-yl)amino]-1-(4-methylpiperidin-1-yl)propan-1-one
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
N3-cyclopentyl-N5-(3-ethoxypropyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4-phenylbutan-2-yl)({2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
2-methyl-2-(4-{1H-[1,2,3]triazolo[4,5-b]pyridin-6-yl}phenyl)propanenitrile
4-{[1-(3-chloro-4-fluorophenyl)-1H-1,2,4-triazol-5-yl]methyl}piperazin-2-one
ethyl 2-{methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}-1,3-oxazole-4-carboxylate
5-(1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-methyl-1,2-oxazole
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
6-(3-chlorophenyl)-N-[2-(1,3-thiazol-4-yl)ethyl]imidazo[2,1-b][1,3]thiazole-3-carboxamide
1-ethyl-4-{[methyl({[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}pyrrolidin-2-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1-(2-phenylethyl)piperazin-2-yl}ethan-1-ol
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-2,5,6-trimethylpyrimidin-4-amine
7-(propan-2-yl)-2-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]-N-(2,3,4-trifluorophenyl)acetamide
1-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-5-methyl-5-phenylpiperidin-2-one
1-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-7-yl]-3-(thiophen-3-yl)propan-1-one
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]amine
(3S,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-{5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-indazol-1-yl)ethan-1-one
9-[(2R)-2-amino-2-phenylacetyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
5-[2-(aminomethyl)-7-fluoro-2,3-dihydro-1-benzofuran-5-yl]pyrazin-2-amine
2-amino-4-(2-methoxyquinolin-3-yl)-6-(pyridin-2-yl)pyridine-3-carbonitrile
2-(2-{[(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}phenoxy)acetamide
N-(2,3-dihydroxypropyl)-5-(2-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(2-methoxyethyl)-3-[1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazol-2-yl]propanamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(2-methylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{1-[(6-methoxypyridin-3-yl)methyl]azetidin-3-yl}morpholine
3-[5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
4-[4-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperazin-1-yl]quinazoline
5-(3-chloro-4-fluorobenzoyl)-1-(cyclopropylmethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{7-hydroxy-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]propanamide
N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}imidazo[1,2-a]pyrimidine-2-carboxamide
2-cyclopropyl-4-phenyl-9-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-1-yl}pyrazine
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(2-methoxyphenyl)propanamide
N-(2-{5-[(cyclohexylmethyl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}ethyl)-4-fluorobenzamide
(3R,5S)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}butanamide
1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-3-(pyridin-3-yl)propan-1-one
3,3,3-trifluoro-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-[(2-fluorophenyl)methyl]-N-[3-(2-methoxyphenyl)propyl]-6-oxopiperidine-3-carboxamide