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1-(4-fluorophenyl)-N-[2-(pyrrolidine-1-sulfonyl)ethyl]cyclopropane-1-carboxamide
N-(3-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}phenyl)butanamide
2-acetyl-8-[(1-propyl-1H-imidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{[4-(3,4-dimethylphenoxy)phenyl]methyl}-3-(hydroxymethyl)pyrrolidin-3-ol
9-[(3-chloro-2-fluorophenyl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(8-{[4-(2-hydroxyethoxy)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]benzamide
4-(5-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl)morpholine
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-(4-methyl-1,4-diazepan-1-yl)ethan-1-one
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazine-2-carboxamide
6-cyano-N-[(3R,4S)-4-cyclopropyl-1-[3-(methylsulfanyl)propyl]pyrrolidin-3-yl]pyridine-3-carboxamide
benzyl(methyl)({3-[4-(propan-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)amine
1-{5-[(4-cyclohexylpiperazin-1-yl)methyl]-2-methoxyphenoxy}-3-(piperidin-1-yl)propan-2-ol
(1S,5R)-3-(1,4-dithiepan-6-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-methoxyphenoxy)acetamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-oxo-2-phenylacetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}({[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl})methylamine
N-[(2-chloropyridin-3-yl)methyl]-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
5-ethyl-N,2-dimethyl-N-[2-(pyridin-4-yl)ethyl]pyrimidin-4-amine
3-[1-(cyclohexylmethyl)-1H-pyrazol-5-yl]-1-(1H-1,2,3,4-tetrazol-5-ylmethyl)urea
1-cyclohexyl-N-cyclopropyl-5-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-[4-(methoxymethyl)piperidin-1-yl]-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridine
(3S,4S)-1-(benzenesulfonyl)-4-[methyl({[3-(trifluoromethyl)phenyl]methyl})amino]pyrrolidin-3-ol
6-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
1-(5-chloropyridin-2-yl)-4-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperazine
5-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
1-[4-(piperidin-1-yl)benzoyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-({4-[4-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)phenol
5-{3-[5-(2-fluoro-4-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}-1H-1,2,3,4-tetrazole
4-amino-3-hydroxy-N-methyl-N-[(4-phenoxyphenyl)methyl]butanamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3,5-dihydroxy-4-methylbenzamide
1-{1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-yl}azetidin-3-ol
[(5-fluoro-1H-indol-2-yl)methyl](methyl)[(5-methyl-1,2-oxazol-3-yl)methyl]amine
1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-4-(pyridin-2-yl)piperazine
N-(2-{[2-(morpholin-4-yl)ethyl]carbamoyl}phenyl)-6-oxo-1,6-dihydropyridine-2-carboxamide
N-methyl-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
(3aR,6aR)-2-(2-hydroxyethyl)-5-[2-(2-oxopiperidin-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 1-(3-{5-[2-(3-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanoyl)piperidine-2-carboxylate
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-(1H-imidazol-4-yl)-1-(3-methylbutyl)-4-phenyl-1H-imidazole
{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
2-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)pyrrolidin-3-yl]benzoic acid
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyrrolidin-3-yl)acetamide
5-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(2-aminopyrimidin-5-yl)methyl]-1-cyclopentyl-N-methyl-6-oxopiperidine-3-carboxamide
(1-benzofuran-2-ylmethyl)(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
3-(2-methoxyphenyl)-N-{[4-(oxolan-2-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)propanamide
N-(butan-2-yl)-N-[(3-chlorophenyl)methyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-cyclohexanecarbonyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-(cyclohexylmethyl)-N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-6-oxopiperidine-3-carboxamide
N-(2-methoxyphenyl)-1-{2-[3-(3-methoxyphenyl)propanamido]ethyl}-1H-1,2,3-triazole-4-carboxamide