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4-(4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}piperidin-1-yl)-2-[1-(1,3-thiazol-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl 2-chloro-4-{[4-(dimethylamino)azepane-1-carbonyl]amino}benzoate
4-[(4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperazin-1-yl)sulfonyl]morpholine
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-3-[(3-fluorophenyl)methyl]-N-methyl-1,2-oxazole-5-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-(5,6-dimethylpyrimidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-N-methylthiophene-2-carboxamide
N-cyclohexyl-3-({[2-(methylsulfanyl)phenyl]carbamoyl}amino)propanamide
2-[methyl({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]ethan-1-ol
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-{[4-(propan-2-yl)phenyl]methyl}pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-{4-[2-(2-methoxyphenyl)acetamido]-1H-pyrazol-1-yl}acetamide
N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-(methylsulfanyl)benzamide
8-[(8-methylquinolin-5-yl)methyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1R,7S)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(3-cyanopyridin-2-yl)piperidine-4-carboxylic acid
3-(but-2-yn-1-yl)-5-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-5-(3-phenylpropyl)imidazolidine-2,4-dione
N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
(4-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}morpholin-2-yl)methanamine
4-[6-(2,4-dichlorophenyl)pyridazin-3-yl]thiomorpholine
2-(cyclopropylmethyl)-8-(1H-1,2,4-triazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(4-methoxy-3,5-dimethylphenyl)-4-(pyridin-4-yl)piperazine-1-carboxamide
2-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1,2-oxazolidin-4-ol
N-cyclopropyl-6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridazin-3-amine
3-(oxolan-3-yl)-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1,2,4-oxadiazole
2-(pent-2-yn-1-yl)-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
[(2S,6S)-4-(1,2-oxazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-(methoxymethyl)-N-methyl-1,3,4-oxadiazole-2-carboxamide
N-[4-(5-chlorothiophen-2-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]butanamide
{3-[(4-fluorophenyl)methyl]-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl}methanol
[(3R,4R)-1-(pyrimidin-2-yl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-[2-(prop-2-en-1-yloxy)phenyl]-1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazole
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-3-(2-phenylpropyl)-1,2-oxazole-5-carboxamide
2,2-dimethyl-N-{[7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}propanamide
2-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
5-{2-[6-(dimethylcarbamoyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-yl]acetamido}pentanoic acid
2-(5-fluoro-2-methoxyphenyl)-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetic acid
6-(2,5-dimethylfuran-3-yl)-N-[(2R)-1-hydroxybutan-2-yl]-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{4-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
[1-ethyl-3-(3-fluorophenoxymethyl)-1H-1,2,4-triazol-5-yl](4-methoxyphenyl)methanol
N3-ethyl-N1-[3-methoxy-5-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-1,3-dicarboxamide
methyl[(3-methylquinoxalin-2-yl)methyl][3-(1H-pyrazol-1-yl)propyl]amine
(1S,5R)-3-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
3-fluoro-N-{3-[(furan-2-ylmethyl)sulfanyl]propyl}-7-methylimidazo[1,2-a]pyridine-2-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
N-[1-(pyrimidin-2-yl)piperidin-3-yl]-2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carboxamide
5-ethyl-4-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}pyrimidin-2-amine
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[3-(propan-2-yloxy)phenyl]methyl}pyrrolidin-3-yl]methanol
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-cyclopropyl-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-methyl-4-(4-{4-[(methylsulfanyl)methyl]piperidine-1-carbonyl}phenyl)butan-2-ol