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9-(2,1,3-benzoxadiazol-5-ylmethyl)-3-cyclopropanecarbonyl-3,9-diazaspiro[5.6]dodecane
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-1-(1-phenylethyl)-1H-1,2,3,4-tetrazole
5-({[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)-2-hydroxybenzoic acid
2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(oxan-4-ylmethyl)acetamide
3-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetamide
N-cyclopropyl-1-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}piperidine-3-carboxamide
4-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}benzonitrile
4-(4-chlorophenyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}butanamide
1-(4-chloronaphthalen-1-yl)-3-{[1-(2-methoxyethyl)-5-oxopyrrolidin-3-yl]methyl}urea
4-(2-chloro-6-fluorophenyl)-N,6-dimethyl-2-oxo-N-(pyrazin-2-ylmethyl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
methyl[1-(1,3-thiazol-2-yl)ethyl]{[3-(1H-1,2,4-triazol-5-yl)phenyl]methyl}amine
methyl[(3-methyl-1H-indol-2-yl)methyl]{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N2-(1-benzylpyrrolidin-3-yl)-N1-(pyridin-3-yl)ethane-1,2-diamine
1-ethyl-6-{[2-(pyridin-3-yl)morpholin-4-yl]methyl}-1H-indole
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-phenylcyclopentyl)methyl]acetamide
(4aS,8aR)-6-[(4-fluorophenyl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
9-[(4-methoxyphenyl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-methylacetamide
N,N-diethyl-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-amine
N-(3-hydroxypropyl)-4-{[(5-methylpyrazin-2-yl)methyl]sulfamoyl}benzamide
N-ethyl-3-[(2-fluorophenyl)formamido]-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
(5S,9aS,9bS)-5-(5-methylfuran-2-yl)-2-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-benzyl-N-[(1R,3S,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl]oxane-2-carboxamide
2-{2-[4-(1,7-dimethyl-1H-indole-2-carbonyl)piperazin-1-yl]ethoxy}ethan-1-ol
N-methyl-3-(1,2-oxazolidin-2-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
7-{[3-(2-methylphenyl)phenyl]methyl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
3-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(2R,6S)-4-[1-(1-cyclohexyl-1H-1,2,3-triazole-4-carbonyl)piperidin-4-yl]-2,6-dimethylmorpholine
3-({[2-(benzyloxy)ethyl]amino}methyl)pyrrolidin-3-ol
N-cyclopentyl-5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-{4-[({[2-(2-methylphenoxy)pyridin-3-yl]methyl}amino)methyl]phenyl}acetamide
[(3-{[(2S,5R)-5-(morpholin-4-ylmethyl)oxolan-2-yl]methyl}phenyl)methyl](prop-2-en-1-yl)amine
1-[3-(2-methyl-1,3-thiazol-4-yl)phenyl]-N-(thiolan-3-yl)piperidin-4-amine
3-{1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
N,8-dimethyl-2-propyl-N-(pyridin-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-methanesulfonyl-N-{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-amine
methyl 4-{[methyl(quinolin-5-ylmethyl)amino]methyl}thiophene-2-carboxylate
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1,2,5-thiadiazole-3-carboxamide
N-{[8-(cyclohexylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
3-(4-methoxy-2-methylbenzoyl)-N,N-dimethylpiperidine-1-sulfonamide
4-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]butanoic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,3,5-trimethyl-1H-pyrazole-4-carboxamide
2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}thiophene-3-sulfonamide
2-[(5-methylpyrazin-2-yl)methyl]-8-(6-methylpyridine-3-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(3-cyclopentylpropyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol