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(3R,9R)-11-(2,5-difluorobenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
5-(2-chlorophenyl)-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]furan-2-carboxamide
N1-(5-methylpyridin-2-yl)-N3-[4-(trifluoromethyl)pyrimidin-2-yl]propane-1,3-diamine
4-chloro-N-{[1-(hydroxymethyl)cyclopentyl]methyl}-2-methylbenzamide
benzyl(butyl)({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N,1,3-trimethyl-N-[2-(1H-pyrazol-4-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-({4-methyl-5-[1-(3-methylpyrazin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)piperidin-4-ol
5-cyclopropanecarbonyl-1'-(3-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-{5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-1H-pyrazole-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[({2-[2-hydroxy-3-(pyrrolidin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]ethyl}acetamide
N-[2-(methylsulfanyl)ethyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
[3-(1-phenylpiperidin-4-yl)-9-propyl-3,9-diazaspiro[5.5]undecan-1-yl]methanol
3-{[4-ethyl-5-oxo-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]methyl}-N,N-dimethyl-1,2,4-oxadiazole-5-carboxamide
1-[3-({[(1-cyclohexylpiperidin-3-yl)methyl](pyridin-3-ylmethyl)amino}methyl)phenyl]ethan-1-one
4-(1H-pyrazol-4-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
3-propyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
1-[4-(2-amino-6-methylpyrimidin-4-yl)piperazin-1-yl]-3-(3,5-dimethylphenyl)propan-1-one
(3R,4R)-1-(9H-fluoren-2-ylmethyl)-4-(4-hydroxypiperidin-1-yl)piperidin-3-ol
3-hydroxy-3-({methyl[(3-methylpyridin-2-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
1-[(2-fluorophenyl)methyl]-N-({8-methylimidazo[1,2-a]pyridin-2-yl}methyl)-6-oxopiperidine-3-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
6-[(3-chloro-4-hydroxyphenyl)methyl]-1-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-3-(2-methylphenyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
8-(2-methoxypyrimidine-5-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-benzyl-N-methyl-3-{1-[2-(pyridin-4-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
5-(5-phenoxyfuran-2-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
3-(3,4-dimethoxybenzoyl)-1-[(2-ethoxyphenyl)methyl]piperidine
6-[(diethylamino)methyl]-N-[4-(methylsulfanyl)phenyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-(2-propoxyethyl)piperazine
N-(cyclopent-3-en-1-yl)-2-methyl-7-(4-methyl-1H-pyrrole-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}quinolin-4-ol
7-(cyclohexylmethyl)-2-cyclopentanecarbonyl-2,7-diazaspiro[4.5]decane
1-{4-[4-(4-methoxybenzoyl)piperazine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-{4-[5-(hydroxymethyl)furan-2-yl]-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl}pyridine-3-carboxamide
methyl 2-(1H-imidazol-2-ylformamido)-2-(3-methylphenyl)acetate
[(3aS,6aS)-2-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)-octahydrocyclopenta[c]pyrrol-3a-yl]methanol
5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-methyl-1H-1,2,4-triazole
3-fluoro-N-[(7-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzamide
4-{2-[(6-phenylpyridazin-3-yl)oxy]hex-5-en-1-yl}thiomorpholine
[(3R,4R)-1-(3,5-difluorobenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
N3-methyl-N3-[3-(3-methylphenoxy)propyl]piperidine-1,3-dicarboxamide
1-(benzyloxy)-8-[2-(thiophen-2-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-(3-{4-[(oxolan-3-yl)amino]piperidin-1-yl}phenyl)-4-phenylbutanamide
4-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-benzyl-N-methyl-3-[1-(6-oxo-1,6-dihydropyridine-2-carbonyl)piperidin-4-yl]propanamide
4-(1H-imidazol-1-yl)-1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxylic acid
N-({5-cyclobutanecarbonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,2-dimethyloxane-4-carboxamide
(5S,9aS,9bS)-5-(6-chloro-2H-chromen-3-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(2S,4S)-N,N-diethyl-1-(2-methoxyacetyl)-4-[2-(3-methyl-1H-pyrazol-1-yl)acetamido]pyrrolidine-2-carboxamide
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl})amine