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4-[(furan-2-ylmethyl)amino]-5-methyl-N-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
3-(2H-1,3-benzodioxole-5-carbonyl)-1-[(5-ethylfuran-2-yl)methyl]piperidine
N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-2-(4-propanoylphenoxy)acetamide
N-[(3S,5S)-1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1H-pyrrole-3-carboxamide
1-(1,4-dioxane-2-carbonyl)-4-(diphenylmethyl)piperazine
1-butyl-5-{[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(3-fluorophenyl)acetyl]piperidin-4-yl}propanamide
N-ethyl-1-(methoxymethyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]cyclobutane-1-carboxamide
N-methyl-N-[1-(4-{[(3-methylthiophen-2-yl)methyl]amino}benzoyl)pyrrolidin-3-yl]acetamide
4-[(2-chlorophenyl)methyl]-1-[2-(2,3-difluorophenyl)acetyl]-1,4-diazepan-5-one
N-(butan-2-yl)-4-(5-{[(2-chlorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidine-1-carboxamide
N-[(3-fluorophenyl)methyl]-9-methoxy-3-[2-(4-methylphenoxy)acetyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
4-[(3-methyl-1H-pyrazol-5-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[5-(1H-pyrrole-2-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
6-[(diethylamino)methyl]-N-(5-fluoro-2-methylphenyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
(5S,9aS,9bS)-5-(2-butyl-1H-imidazol-4-yl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2-ethoxyethyl)-N-(oxan-4-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[(4-fluorophenyl)formamido]-N-{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}propanamide
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}pyrrolidin-3-yl]acetamide
N4-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-5,6-dimethylpyrimidine-2,4-diamine
2-{4-[3-(4-benzylpiperidin-1-yl)-3-oxopropyl]piperidin-1-yl}acetamide
3-(2,5-dimethoxyphenyl)-1-(2-methylfuran-3-carbonyl)pyrrolidine
2-[4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazin-1-yl]ethan-1-ol
8-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-[(5-butylthiophen-2-yl)methyl]-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
ethyl 2-{1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]piperidin-2-yl}acetate
2-{2-[1-(4-fluorobenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
(3R,4R)-1-(2,5-dimethoxybenzoyl)-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}benzamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)furan-2-carboxamide
1-(oxan-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
1-{3-[2-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(trifluoromethyl)pyrimidin-4-amine
2-[3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
(2S,4R)-4-amino-N-methyl-1-{4-[(pyridin-4-ylmethyl)amino]benzoyl}pyrrolidine-2-carboxamide
N,N-dimethyl-3-[(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)sulfamoyl]benzamide
(5S,9aS,9bS)-5-phenyl-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1,9-dioxaspiro[5.5]undecan-4-amine
1-(2-ethylphenyl)-3-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
7-methyl-2-{[2-methyl-5-(1,2-oxazol-5-yl)furan-3-yl]sulfonyl}-2,7-diazaspiro[4.5]decan-6-one
6-oxo-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-1-(2-phenylethyl)piperidine-3-carboxamide
2-methoxy-N,N-bis(propan-2-yl)-6-[2-(propanamidomethyl)phenyl]benzamide
6-oxo-N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}-1,6-dihydropyridine-3-carboxamide
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[2-(1,3-thiazol-4-yl)ethyl]urea
7-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
methyl 2-{[(cyclooctylcarbamoyl)methyl]amino}-3-hydroxypropanoate
methyl (2S,4R)-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]-1-{[4-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxylate
2-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
(2R,4S)-1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-4-hydroxypiperidine-2-carboxylic acid