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methyl 2-[(2-methoxyethyl)sulfamoyl]-6-{[3-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)sulfonyl]-3-(3-chlorobenzoyl)piperidine
N-benzyl-N-methyl-2-(4-methylpiperazine-1-carbonyl)-2,3-dihydro-1H-inden-2-amine
7-(4-chloro-1H-pyrazole-3-carbonyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(pyridin-4-yl)pyrimidin-2-amine
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]pyrrolidine-2-carboxamide
5-[1-ethyl-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1H-pyrrole-3-carbonitrile
1-({5-[(3-fluoro-4-methoxyphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-[2-(3-methoxyphenyl)phenyl]-1-(3-phenylbutyl)piperidine-4-carboxamide
4-{4-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
(E)-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-2-phenylethene-1-sulfonamide
3-{[(5-methyl-1,2-oxazol-3-yl)methyl]sulfamoyl}-N-(oxolan-3-ylmethyl)benzamide
{2-[(1H-1,3-benzodiazol-2-ylmethyl)[(5-methylthiophen-2-yl)methyl]amino]ethyl}dimethylamine
2-(methylamino)-N-({1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
3-butanamido-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]benzamide
1-(2-chloro-5-fluorophenyl)-3-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]urea
2-(3-methoxypropyl)-8-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
1-[3-(2-methylpyrimidin-4-yl)phenyl]-N-[1-(pyridin-3-yl)propan-2-yl]piperidin-4-amine
4-(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)-N-(furan-2-ylmethyl)piperidine-1-carboxamide
2-(2-aminoethyl)-5,6-dimethyl-N-[1-(pyridin-3-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
5-(7-fluoro-2-methylquinoline-4-carbonyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-methyl-6-({4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
5-(2-chlorophenyl)-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]furan-2-carboxamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-1-ethylpiperidin-3-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-({5,7-dimethylimidazo[1,2-a]pyridin-2-yl}methyl)acetamide
3-[4-(3,6-dimethylpyrazin-2-yl)piperazine-1-carbonyl]-2-methyl-1,2,3,4-tetrahydroisoquinoline
6-{3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one
5-methyl-N-({1-[(E)-2-phenylethenesulfonyl]piperidin-3-yl}methyl)-1,2-oxazole-3-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,3-dimethylfuran-2-carboxamide
3-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-3-methyl-1-phenylurea
N-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,4,5-trifluorobenzamide
N3-methyl-N5-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3-dihydro-1H-imidazol-2-one
4-(4-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]amino}piperidin-1-yl)-6-ethyl-N,N-dimethylpyrimidin-2-amine
2-methyl-3-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-2,8-diazaspiro[4.5]decane
methyl 1-[5-(ethylcarbamoyl)-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carbonyl]piperidine-2-carboxylate
ethyl 4-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)piperazine-1-carboxylate
5-{[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-methyl-N-(thiophen-2-ylmethyl)piperidine-4-carboxamide
5-(3-fluorophenyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1,2,4-triazin-3-amine
5-[(2,5-dimethoxyphenyl)methyl]-4-(thiophen-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
3-{[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-methyl-N-{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoethyl}propanamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}benzamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-4-(4-oxo-3,4-dihydroquinazolin-3-yl)butanamide
1-({4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)-4-(pyridin-3-yl)piperidin-4-ol
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide