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dimethyl(3-{3-[3-(pyridin-3-yl)phenyl]-1H-pyrazol-1-yl}propyl)amine
ethyl 5-{[(butan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-(quinolin-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[4-({[2-(methylsulfanyl)ethyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
4-chloro-5-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
N-({7-[2-(4-chloro-2-methylphenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)cyclopropanecarboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-{5-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-yl}piperazine
5-{[(3-methoxyphenyl)methyl]amino}-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{1-[6-(2-fluoro-6-methoxyphenyl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
ethyl 4-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)piperazine-1-carboxylate
5-(1-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propanoyl}pyrrolidin-2-yl)thiophene-2-carboxamide
8-[(2-chlorophenyl)methyl]-1-ethyl-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3-chloro-4,5-dimethoxyphenyl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
1-cycloheptyl-N-methyl-N-[2-(4-methylphenoxy)ethyl]-6-oxopiperidine-3-carboxamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(naphthalene-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
5-(1-cyclopentanecarbonylpiperidin-4-yl)-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
2-methyl-N-({3-methyl-7-[2-(pyrrolidin-1-yl)acetyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-1,3-thiazole-4-carboxamide
N-{4-[(7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenyl}acetamide
1-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propan-1-one
5-methyl-5-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-4-hydroxy-2-(pyridin-4-yl)pyrimidine-5-carboxamide
6-oxo-N-(1-phenylpiperidin-4-yl)-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
(2S,3R)-2-amino-1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-hydroxybutan-1-one
5-(propan-2-yl)-4-[3-(pyridin-3-yl)azetidin-1-yl]pyrimidine
1-(3-chloro-2-methylbenzenesulfonyl)-4-[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
3-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidine-1-carbonyl]-6-methoxy-1,4-dihydroquinolin-4-one
N-methyl-1-[3-(morpholin-4-yl)propyl]-6-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-3-carboxamide
3-[1-(2,6-dimethoxypyrimidine-4-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-methyl-1,4-dihydroquinolin-4-one
N-(4-methoxyphenyl)-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}acetamide
N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
N-{1-[1-(2-acetamido-3-methylbutanoyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-N-methyl-2-(1H-pyrazol-1-yl)acetamide
N-cyclopropyl-1-{1-[4-(trifluoromethyl)benzoyl]piperidin-4-yl}piperidine-4-carboxamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]pyrrolidin-3-yl]methanol
1-methyl-2-oxo-8-[(3-phenylphenyl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-2-(2,5-dioxoimidazolidin-4-yl)acetamide
3-benzyl-1-(2-methyl-5-propylpyrimidin-4-yl)piperidine-3-carboxylic acid
4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}-1λ6-thiomorpholine-1,1-dione
2-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-4H-chromen-4-one
{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(3-methylpyridin-4-yl)methyl]acetamide
N,3-dimethyl-N-(oxan-2-ylmethyl)-1-propyl-1H-pyrazole-4-carboxamide
{4-[(4-chlorophenyl)methyl]-1-(3-fluoropyridin-2-yl)piperidin-4-yl}methanol
2-fluoro-4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenol
1-(cyclohexylmethyl)-3-hydroxy-3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}piperidin-2-one
N-[(2-methoxyphenyl)methyl]-2-(2-methylphenyl)-N-(pyridin-3-ylmethyl)acetamide
6-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]hexan-1-ol
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1,3-benzoxazole