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N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}thiophene-2-carboxamide
5-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
5-(methoxymethyl)-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)thiophene-2-carboxamide
6-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
(3S,4S)-3-(dimethylamino)-4-hydroxy-N-[2-(3-methylphenyl)-1,3-benzoxazol-6-yl]pyrrolidine-1-carboxamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
4-{[3-(dimethylamino)-2,2-dimethylpropyl]amino}pyrimidine-5-carboxylic acid
1-(3-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
4-(2-ethoxyacetyl)-1-(2-phenylphenyl)piperazin-2-one
methyl 6-[4-(2-methylphenoxy)piperidin-1-yl]pyrimidine-4-carboxylate
benzyl (7S,9aR)-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
3-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-N,N-dimethylpropane-1-sulfonamide
(1S,5R)-6-methyl-3-(2-phenoxybenzoyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(6-aminopyridine-3-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(3S,4R)-1-(3-methyl-1,2-oxazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-cyclopentyl-2-[(3-fluorophenyl)methyl]morpholine
3-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-2-methyl-1,8-naphthyridine
5-methyl-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[3-(2-chlorophenoxy)azetidin-1-yl]-2-ethoxyethan-1-one
8-(3-fluoro-4-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-methyl-N-(2-phenylethyl)-1-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[3-(1H-imidazol-1-yl)propyl]-3-(1-oxo-2,3-dihydro-1H-inden-5-yl)urea
1-[(2-chlorophenyl)methyl]-4-[(2-methyl-5-propylpyrimidin-4-yl)amino]pyrrolidin-2-one
N-[1-(butan-2-yl)-3-methyl-1H-pyrazol-5-yl]-2-[4-(3-methoxypyridin-2-yl)-1H-pyrazol-1-yl]acetamide
3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)-5-[1-(thiophene-3-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-[(2-chloro-4-fluorophenyl)methyl]-N-[2-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{3-[4-(4-chlorophenyl)piperazin-1-yl]-3-oxopropyl}-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
1-methyl-N-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-3-propyl-1H-pyrazole-5-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-(4-fluorophenyl)-4-[1-(2,4,5-trifluorobenzoyl)piperidin-3-yl]piperazine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(methylsulfanyl)propanamide
2-({4-[(8-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperazin-1-yl}methyl)benzonitrile
(4aR,8aR)-2-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[2-(3-phenylpropyl)morpholin-4-yl]-3-(pyridin-4-yl)propan-1-one
2-{1-[(6-methyl-2H-1,3-benzodioxol-5-yl)methyl]piperidin-2-yl}acetic acid
2-chloro-4-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)phenol
9-methoxy-N-methyl-7-oxo-3-(1-phenylcyclopropanecarbonyl)-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]-5-(propan-2-yl)pyrimidine
5-acetyl-6-methyl-3-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-ethyl-6-(4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyrimidine
N-({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-2-(2-methoxyphenoxy)acetamide
N-[2-(2-oxopiperidin-1-yl)ethyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
N-[(3,4-dimethoxyphenyl)methyl]-2,2-diphenyl-N-(pyridin-2-ylmethyl)acetamide
1-(4-benzylpiperazin-1-yl)-3-[1-(4,4,4-trifluorobutyl)piperidin-3-yl]propan-1-one
N-{[7-(2,4-dimethylbenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
(1R,5S)-3-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-methyl-4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-1-(4-methylphenyl)piperazin-2-one