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N-[(5-methylpyrazin-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-methyl-N-({8-propyl-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-pyrazole-5-carboxamide
N-[3-(furan-2-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-4-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-(4,6-dimethoxypyrimidin-2-yl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-(1-{4-[4-(2-fluorophenyl)piperazine-1-carbonyl]phenyl}-1H-pyrazol-4-yl)oxolane-3-carboxamide
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
(1S,6R)-9-(5-amino-4-phenyl-1H-pyrazole-3-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(cyclohex-1-en-1-yl)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methylacetamide
1-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-2-(2H-indazol-2-yl)ethan-1-one
8-[2-(4-fluorophenoxy)acetyl]-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-aminoethyl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-(piperidin-4-ylmethyl)-3-[4-(1H-pyrazol-4-yl)phenyl]urea
[(5-chloro-1H-indol-2-yl)methyl]({[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
methyl (2S,4S)-1-[(3-fluorophenyl)methyl]-4-propanamidopyrrolidine-2-carboxylate
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-methyl-2-(morpholin-4-yl)propyl]acetamide
[1-(benzenesulfonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
N-[1-({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)piperidin-4-yl]acetamide
1-[(2-fluorophenyl)methyl]-N-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperidin-3-amine
4-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-cyclohexyl-3-hydroxy-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(pyridin-4-yl)ethyl]-1,3-benzoxazole-6-carboxamide
2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
2-{1-[(5-methylfuran-2-yl)methyl]-4-{[1-(propan-2-yl)-1H-indol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
N-[(7-{[5-(3-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]-2-(3-fluorophenyl)acetamide
1-[4-(2-methoxyethyl)piperazin-1-yl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propan-1-one
(3S,4S)-1-{[4-(carbamoylmethoxy)-3-chlorophenyl]methyl}-4-cyclopropylpyrrolidine-3-carboxylic acid
2-(diethylamino)-N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
1-[3-(2-methoxyethoxy)phenyl]-3-[1-(thiophen-3-yl)ethyl]urea
4-{1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
(3R,4S)-4-[methyl({[3-(2-methylphenyl)phenyl]methyl})amino]oxolan-3-ol
2-(4-{3-[(3-ethylphenyl)carbamoyl]propanamido}piperidin-1-yl)acetic acid
3-({[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)amino}methyl)benzoic acid
1-(2-methyl-1,3-thiazole-4-carbonyl)-3-phenylpiperazine
2-[2-(dimethylamino)phenyl]-N-(propan-2-yl)pyridine-4-carboxamide
N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]thiophene-2-carboxamide
(2-{[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl][(3-methylthiophen-2-yl)methyl]amino}ethyl)dimethylamine
5-cyclopropyl-N-(2,2-dimethyloxan-4-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-methyl-3-phenyl-8-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,8-diazaspiro[4.5]decan-2-one
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)acetamide
1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]-2-(4-methylphenoxy)ethan-1-one
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
ethyl 2-(4-{[3-(naphthalen-1-yl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetate
5-[1-(3-chlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-phenylpropyl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-5-carboxamide
1-{1-[5-(propan-2-yl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl]piperidin-4-yl}piperidin-4-ol
1-[(4aS,8aR)-4a-(hydroxymethyl)-6-(pyrimidin-2-yl)-decahydro-1,6-naphthyridin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
1-(carbamoylmethyl)-N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]piperidine-4-carboxamide
5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-[1-(3-phenylpropanoyl)piperidin-4-yl]imidazolidine-2,4-dione
4-(4-methylphenyl)-5-(pyrimidin-5-yl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidin-2-amine