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3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidine
2-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
2-methoxy-N-[(3S)-2-oxoazepan-3-yl]-N-({4-[3-(pyridin-3-yl)propoxy]phenyl}methyl)benzamide
6-methyl-2-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl](methyl)[3-(phenylsulfanyl)propyl]amine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](2-methylpropyl)(pyridin-2-ylmethyl)amine
3-[(3R,4S)-3-amino-4-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(oxolan-2-yl)-N-propylthiophene-2-carboxamide
5-[(3-cyclopropyl-1H-1,2,4-triazol-5-yl)methyl]-3-phenyl-1H-1,2,4-triazole
2-[(2-chlorophenyl)methyl]-4-[3-(morpholine-4-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
[4-(2-phenoxyethyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl]methanol
(1S,2S)-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-1-phenylpropane-1,3-diol
2-{4-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-1-(4-methylpiperidin-1-yl)ethan-1-one
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-2-carboxamide
4-{1-[(2-chloro-4,5-dimethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
dimethyl[2-(2-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-yl}-1H-imidazol-1-yl)ethyl]amine
3-{[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}piperidin-3-ol
1-(5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl)pyrrolidine
N-{2-ethyl-5-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1-methyl-1H-1,3-benzodiazol-7-yl}-2-methoxybenzamide
N-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-yl}pyridin-2-amine
4-{[4-(difluoromethoxy)phenyl]methyl}-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl)ethan-1-ol
N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
ethyl(methyl){[5-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amine
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-6-(trifluoromethyl)pyridine
N-(1-{1-[(2S)-2-acetamidopropanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
6-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]pyridine-3-carboxylic acid
4-[(4-methoxyphenyl)methyl]-1-(5-methylthiophene-2-carbonyl)-1,4-diazepan-5-one
2-(2-chloro-6-fluorobenzamido)-7-oxo-N-[1-(thiophen-3-yl)propan-2-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
1-{2-[1-(pent-4-enoyl)piperidin-2-yl]ethyl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-{4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}pyridine-4-carboxamide
3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
1-[(3S,4R)-4-hydroxy-4-methyl-3-(2-methylpropyl)piperidin-1-yl]-4-(4-methoxyphenyl)butan-1-one
3-cyclopropyl-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)-1H-pyrazole-5-carboxamide
2-(2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindole-1,3-dione
(3S,4R)-4-(2-methylphenyl)-1-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
(2S,4R)-4-amino-1-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-methylpyrrolidine-2-carboxamide
2-(1,3-benzoxazol-2-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
N-[(3-methylphenyl)methyl]-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
1-benzyl-5-(cyclopropylamino)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N2-cyclopentyl-N2-[(3-methylthiophen-2-yl)methyl]pyrrolidine-1,2-dicarboxamide
2-{1-methyl-4-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(1R,5R)-6-(cyclopropylmethyl)-3-(3-methoxypyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-{2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholin-4-yl}-3-oxopropyl)-6-methyl-1,2-dihydropyridin-2-one
3-[(3R,4S)-1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-2-butyl-1,3-benzoxazole
{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})amine
N-[3-hydroxy-1-(4-methylphenyl)propyl]-4-propylpyrimidine-5-carboxamide
1-(2-methoxyethyl)-8-[(2-methoxyphenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione