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2-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,2-dihydroisoquinolin-1-one
4,5-dimethyl-6-(1H-pyrazol-4-yl)-2-(trifluoromethyl)pyrimidine
(3aS,6aS)-2-(furan-3-carbonyl)-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(3R,4R)-1-[(4,5-dimethylfuran-2-yl)methyl]-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
1-[(2-methylphenyl)methyl]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(benzylsulfanyl)ethyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
N-butyl-3-(1H-1,2,3,4-tetrazol-1-yl)-N-(thiophen-3-ylmethyl)propanamide
2-[(2-{[1-(2,5-dimethoxyphenyl)ethyl]carbamoyl}phenyl)amino]acetic acid
2-(2-methoxyethyl)-8-(4-methylquinolin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
3-phenoxy-1-[3-(pyridin-2-yl)azetidin-1-yl]propan-1-one
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
[1-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperidin-4-yl]methanol
(2S,4R)-4-(dimethylamino)-2-(hydroxymethyl)-N-[4-(trifluoromethoxy)phenyl]pyrrolidine-1-carboxamide
1-{1-[1-(4-chloro-2-methoxybenzoyl)piperidin-4-yl]ethyl}-4-methylpiperazine
1-(5-acetyl-2-ethoxyphenyl)-3-methyl-3-[(5-methylfuran-2-yl)methyl]urea
1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]-4-(thiophene-2-carbonyl)piperazine
8-(5-hydroxypyrazine-2-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[5-(2-methylpropyl)-1H-pyrazol-3-yl]-1H-1,2,3-triazole
3-[(2-methylprop-2-en-1-yl)oxy]-N-{[6-(trifluoromethyl)pyridin-3-yl]methyl}benzamide
(2R,3S,6R)-5-(isoquinolin-5-ylmethyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-N,2,2,6,6-pentamethylpiperidin-4-amine
N-[2-(diethylamino)ethyl]-2-[2-(morpholin-4-ylmethyl)-4-(pyrazin-2-yl)phenoxy]acetamide
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-1-(4-methyl-1,4-diazepan-1-yl)propan-1-one
6-[(3,4-difluorophenyl)methyl]-N-(3,5-dimethylphenyl)-6-azaspiro[2.5]octane-1-carboxamide
4-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1,3-oxazolidin-2-one
7-(2-cyclohexylethyl)-2-(5-ethyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-{2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-[furan-2-yl(phenyl)methyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)piperidin-2-one
2-(2-chlorophenyl)-2-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}acetic acid
2-(2,6-dimethoxy-4-methylphenyl)-2-(4-methyl-1,4-diazepan-1-yl)acetic acid
N-methyl-N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-2-carboxamide
2-methyl-5-{3-[(4-methylpiperazin-1-yl)methyl]piperidine-1-carbonyl}phenol
5-{2,7-dimethylimidazo[1,2-a]pyridin-3-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[2-(3-methoxyphenyl)phenyl]-1-[(2-methylpyrimidin-5-yl)methyl]piperidine-4-carboxamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-4-(3,5-dimethyl-1H-pyrazol-1-yl)benzamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
2-[4-(1-cyclohexylpiperidine-4-carbonyl)piperazin-1-yl]pyrimidine
N-[1-(3-hydroxyadamantan-1-yl)ethyl]-3-[2-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(2,5-dioxoimidazolidin-4-yl)propanamide
N-{[1-(pyridin-4-ylmethyl)piperidin-3-yl]methyl}quinoline-8-sulfonamide
1-(4-benzylpiperazin-1-yl)-3-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}propan-1-one
(2S,4S)-4-amino-1-[(2-fluoro-5-methoxyphenyl)methyl]pyrrolidine-2-carboxylic acid
N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
1-benzyl-N-methyl-5-(pyridin-3-ylmethyl)-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl 1-[(3R,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(propan-2-yl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-[5,6-dimethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
N-{[5-fluoro-7-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(2-methoxyphenyl)propanamide