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4-[(2,4,6-trifluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
ethyl 3-{[1-(3,4-difluorophenyl)piperidin-4-yl]amino}azepane-1-carboxylate
2-phenyl-1-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-yl}ethan-1-ol
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]acetamide
N,N-dimethyl-2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}propanamide
(4aR,7aS)-1-(2-methylpropyl)-4-[3-(pyridin-4-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(4-fluorophenyl)-3-{[3-(5-methylthiophen-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
1-(2-methoxyacetyl)-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-3-carboxamide
1-[3-(2-ethoxyethoxy)benzoyl]-3-(3-methylphenoxy)azetidine
3-(pentan-2-yl)-8-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-4-amine
1-ethyl-N-[(3S,5S)-1-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-yl]piperidin-4-amine
methyl 5-{[(2,3-difluorophenyl)methyl]amino}-3-(furan-2-amido)-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-{2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetyl}-1-(4-methylphenyl)piperazin-2-one
N-(furan-2-ylmethyl)-3-(2-hydroxyphenyl)-N-(prop-2-en-1-yl)propanamide
N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
N-methyl-N-[2-(2-methylphenyl)-1-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}ethyl]-2-(1H-pyrazol-1-yl)acetamide
N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]-2-(thiophen-3-yl)acetamide
1-{2-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-oxoethyl}pyrrolidin-2-one
ethyl 2-(3-methylbutyl)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxylate
N-methyl-2-(pyridin-3-yl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-5-carboxamide
N-butyl-5-methyl-4-[(prop-2-en-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
3-(2-methoxyphenyl)-N-[1-({methyl[(4-phenyl-1,3-thiazol-2-yl)methyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
4-[5-(4-methoxy-4-phenylpiperidine-1-carbonyl)-1H-pyrazol-3-yl]phenol
methyl 2-(4-cyanopyridin-2-yl)benzoate
2-methyl-4-{3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenyl}butan-2-ol
(4aS,7aR)-1-(4-oxo-1,4-dihydroquinoline-2-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[3-(morpholin-4-ylmethyl)phenyl]-2-(pyrrolidin-1-yl)pyrimidin-4-amine
methyl 5-[(7-methoxy-1,2,3,4-tetrahydronaphthalen-2-yl)amino]-1-(2-methoxyethyl)-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[(oxan-4-yl)amino]-1-(2-phenylethyl)pyrrolidin-2-one
3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-ethyl-5-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}pyrimidin-2-amine
3,5-dimethyl-1-(1-{[3-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-yl)-1H-pyrazole
methyl 7-oxo-3-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-9-(propan-2-yloxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
6-(benzyloxy)-4-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
4-[2-(propan-2-yloxy)phenyl]benzamide
ethyl 2-[2-(4-fluorophenyl)morpholin-4-yl]pyridine-3-carboxylate
methyl 1-{3-[4-(azetidin-1-ylmethyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
1-{2-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,2-dihydropyridin-2-one
5-(1-ethylpiperidine-4-carbonyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(3R,4S)-3,4-dimethyl-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-4-ol
4-phenyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]azepane
6-{2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}-5,6,7,8-tetrahydro-1,6-naphthyridine
3-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]propanamide
3-{5-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-ethyl-N-[(5-fluoro-2-methylphenyl)methyl]-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
3-(1-methylpiperidin-3-yl)-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}propanamide
4-benzoyl-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine
4-(3-phenylpiperidine-1-carbonyl)-2-(1H-pyrazol-4-yl)quinoline
5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidin-2-one