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5-[4-(benzyloxy)piperidine-1-carbonyl]-1-(pyridin-2-ylmethyl)piperidin-2-one
(2S,4R)-4-amino-N-ethyl-1-[(1-methyl-1H-imidazol-4-yl)sulfonyl]pyrrolidine-2-carboxamide
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoxaline
3-methyl-1-{[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl}piperidine
6-fluoro-2-({[2-(4-methyl-1H-pyrazol-1-yl)ethyl]amino}methyl)quinolin-4-ol
propan-2-yl N-{2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)morpholin-2-yl]ethyl}carbamate
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
[3-(2-methoxyethyl)-1-{[4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl]methanol
6-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
methyl 1-[5-(phenoxymethyl)-1H-pyrazole-3-carbonyl]-2,5-dihydro-1H-pyrrole-2-carboxylate
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(2-methylphenyl)pyrrolidin-3-ol
N,N-diethyl-2-({4-[(3-hydroxy-4-methoxyphenyl)methyl]-2-oxo-1-(2-phenylethyl)-1,4-diazepan-6-yl}oxy)acetamide
5-benzenesulfonamido-1-ethyl-2-methyl-N-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-1,4-dihydropyridine-3-carboxamide
4-(5-methoxyfuran-2-carbonyl)-1-(2-methylphenyl)piperazin-2-one
[(4-methanesulfonylphenyl)methyl](methyl)(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
N-(2-methyl-1,3-benzothiazol-5-yl)-6-(4-methyl-1,3-oxazole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
1-(2-methyl-1-benzofuran-5-carbonyl)-3-(3-methylphenoxy)azetidine
4-(2,3-dimethoxybenzoyl)-2-[(4-fluorophenyl)methyl]morpholine
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]benzonitrile
N-(1-{7-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)furan-2-carboxamide
(2S,4S)-4-amino-N,1-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyrrolidine-2-carboxamide
3-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
1-(3,5-dimethylphenyl)-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazin-2-one
1-{1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}piperidine-3-carboxylic acid
(4aR,7aS)-1-methyl-4-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-(2-oxoazepan-3-yl)benzamide
methyl (2S)-2-[(1-{4-[2-(3-fluorophenyl)acetamido]phenyl}piperidin-4-yl)amino]-3-methylbutanoate
2-(2-methylpyrrolidin-1-yl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
N-[(3-fluoro-4-methylphenyl)methyl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}acetamide
1-{[4-(2H-1,3-benzodioxol-5-yl)phenyl]methyl}-1H-imidazole
9-[(2-chlorophenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-methyl-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
5-chloro-2-methoxy-4-[1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]pyridine
1-[2,2-dimethyl-3-(pyrrolidin-1-yl)propyl]-4-(4H-1,2,4-triazol-3-yl)piperidine
2-(4-hydroxypiperidin-1-yl)-N-[1-(2-methoxyphenyl)ethyl]-N-methylacetamide
2,5-dichloro-N-{2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}benzamide
7-hydroxy-6-methoxy-4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydroquinolin-2-one
4-[3-(morpholine-4-carbonyl)phenoxy]thiane-4-carboxylic acid
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2,2-dimethylpropan-1-one
3-[2-(azepan-1-yl)-2-oxoethyl]-3-(2-chlorophenyl)-1-(3-methoxypropyl)pyrrolidine-2,5-dione
N-({1-[3-(3-methoxyphenyl)benzoyl]piperidin-4-yl}methyl)acetamide
6-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-N-methyl-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
4-[3-(oxan-4-yl)-5-(1H-pyrrol-2-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
5-ethyl-5-[1-(furan-3-ylmethyl)piperidin-4-yl]-3-[2-(4-methoxyphenyl)ethyl]imidazolidine-2,4-dione
4-(4-methylphenoxy)-N-[1-(pyridin-3-yl)ethyl]piperidine-4-carboxamide
4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-(3-fluorophenyl)piperazin-2-one
2-methyl-1-{[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-1,4-diazepan-5-one
1-cycloheptyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-6-oxopiperidine-3-carboxamide