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5-chloro-N-(2-methoxyethyl)-4,6-dimethyl-2-oxo-N-(pyridin-3-ylmethyl)-1,2-dihydropyridine-3-carboxamide
methyl 1-[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]piperidine-4-carboxylate
1-[(4-ethoxyphenyl)methyl]-1-(2-methoxyethyl)-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
2-amino-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-6-(2-methylpropyl)pyrimidine-4-carboxamide
1-[(2-fluorophenyl)methyl]-5-[4-(pyrrolidin-1-yl)piperidine-1-carbonyl]piperidin-2-one
N-({1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}methyl)-4-fluorobenzamide
N-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-N-methylthian-4-amine
4-(2-acetamidoethoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
1-(4-{2-azaspiro[4.4]nonan-2-ylmethyl}-2-methoxyphenoxy)-3-(diethylamino)propan-2-ol
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-(3-hydroxy-3-phenylpropyl)-N-methyl-1,3-oxazole-4-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-6-(naphthalen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[(diethylcarbamoyl)methyl]-N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-[3-(aminomethyl)pyrrolidine-1-carbonyl]-2-(3,5-dichlorophenyl)pyrimidin-4-ol
N-[(3R,7S,8aS)-3-[(benzylsulfanyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-[1-(pyridin-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-[(4-methylpiperidin-1-yl)methyl]piperidin-2-one
2-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyridin-3-ol
(4aS,8aR)-6-(3-hydroxybenzoyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(2-ethoxypyridin-3-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-(3-methylbutyl)-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
5-benzenesulfonamido-1-ethyl-N-(1-hydroxy-2-methylpropan-2-yl)-2-methyl-1H-1,3-benzodiazole-7-carboxamide
8-(9H-purin-6-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
methyl[(2-methyl-2H-indazol-3-yl)methyl][1-(4-methylpyridin-2-yl)propan-2-yl]amine
2-[1-(2-methoxyphenyl)-5-[(2-methyl-1H-1,3-benzodiazol-5-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
2-cyclopentyl-9-[2-(4-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[3-(propan-2-yloxy)benzoyl]-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
methyl 1-[(3R,5S)-5-(cycloheptylcarbamoyl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
N-(3-fluorophenyl)-3-[4-(1H-pyrazol-1-ylmethyl)piperidin-1-yl]propanamide
1-oxo-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-chloro-N-cyclopropyl-N-({3-[(1-methoxypropan-2-yl)oxy]phenyl}methyl)benzamide
methyl 3-[(2-fluoro-5-methoxyphenyl)methyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(3S,4S)-1-[5-(4-methoxyphenyl)furan-2-carbonyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-methoxy-1-{1'-[3-(5-methylfuran-2-yl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
(3aS,6aR)-5-(1H-imidazol-2-ylmethyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
7-[(4-fluorophenyl)methyl]-2-(thiophene-2-carbonyl)-2,7-diazaspiro[4.5]decane
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-2-yl)ethyl]acetamide
2-[4-({methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}methyl)phenoxy]propanoic acid
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-oxo-2-phenylacetamide
3-{2-[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,2,3-oxadiazol-3-ium-5-olate
[3-benzyl-1-(pyridin-3-ylmethyl)piperidin-3-yl]methanol
5-{1-[(4-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
methyl (2S)-1-({4-[(3,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)pyrrolidine-2-carboxylate
2-butyl-4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
5-[1-(4-methoxybenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-(4-{[1-(cyclohex-2-en-1-yl)-1,2,5,6-tetrahydropyridin-3-yl]methoxy}piperidin-1-yl)-2-methylpropan-1-one
1-(1-ethylpyrrolidine-3-carbonyl)-4-(3-methoxybenzoyl)piperazine
4-[(2,3-dihydro-1-benzofuran-5-ylmethyl)amino]-1-[2-(4-methoxyphenyl)ethyl]pyrrolidin-2-one
1-[2-(hydroxymethyl)piperidin-1-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one