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4-(5-propyl-1,2-oxazole-3-carbonyl)-2-(trifluoromethyl)morpholine
3-{5-methanesulfonyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]pyrimidin-2-amine
[(3-chloropyridin-4-yl)methyl](methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
9-(3-hydroxypyridine-2-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[4-(3-methoxypyrazin-2-yl)morpholin-2-yl]methanamine
1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}-3-(1H-pyrazol-5-yl)piperidine
2-{4-[(3,5-difluorophenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-{[7-chloro-5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,4-dimethyl-1,3-thiazole-5-carboxamide
(1S,5R)-6-(cyclopropylmethyl)-3-(2-methyl-6-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3,7-dimethyl-11-(1,3-thiazole-5-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
(3aS,6aS)-2-(1H-imidazol-2-ylmethyl)-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-[3-(hydroxymethyl)phenyl]-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
2-methoxy-N-(3-methyl-1-{7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)acetamide
5-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-1-ethyl-3-(propan-2-yl)-1H-pyrazole
N-{[7-(2-chloro-6-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2H-1,3-benzodioxole-5-carboxamide
2-methyl-N-[4-(pyridin-2-yl)butyl]imidazo[1,2-a]pyridine-6-carboxamide
7-(cyclohex-3-en-1-ylmethyl)-N-(pyridin-2-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-cyclopropyl-4-{[(3S,4S)-3-hydroxy-4-(propan-2-yloxy)pyrrolidin-1-yl]sulfonyl}benzamide
1-[(2-chlorophenyl)methyl]-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepane
1-(5-fluoro-1-methyl-1H-indole-2-carbonyl)azepan-4-amine
N-cyclopentyl-3-{[(2-methyl-1,3-thiazol-4-yl)methyl]sulfamoyl}benzamide
3-[2-(2-hydroxyethoxy)ethyl]-6,8-dimethyl-3,4-dihydroquinazolin-4-one
N3-cyclohexyl-N5-cyclooctyl-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
1-{3-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
5-{2-[(1R,5S)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
3-(1H-1,3-benzodiazol-1-yl)-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
3-cyclopropyl-1-phenyl-5-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-ylmethyl}-1H-1,2,4-triazole
(2S)-2-{4-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-1,2,3-triazol-1-yl}-3-(pyridin-4-yl)propanoic acid
methyl 4-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}benzoate
N-(3-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-3-oxopropyl)-N-methylmethanesulfonamide
N-[(3S,4R)-1-[2-(2,5-dioxoimidazolidin-1-yl)acetyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
(3S)-1-ethyl-4-[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-methylpiperazin-2-one
4-[5-(pyrimidin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonyl]morpholine
1-{3-[(4-ethyl-1,4-diazepan-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
8-(4-fluoro-2-methylbenzoyl)-5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine
N-methyl-3-(piperazine-1-sulfonyl)-N-(pyrazin-2-ylmethyl)benzamide
N-butyl-3-({[(2,2-dimethyl-1-phenylcyclopropyl)methyl]amino}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decane
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-5-methoxy-1,4-dihydropyridin-4-one
4-[(2R,6S)-2,6-dimethylpiperidine-1-carbonyl]-7-methyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
4-[2-(methoxymethyl)piperidine-1-carbonyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine
methyl 5-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-methyl-3-(4H-1,2,4-triazol-4-yl)benzamide
1'-(8-chloroquinolin-2-yl)-5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 1-[2-(1H-indol-3-yl)ethyl]-5-{[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]amino}-3-(3-methoxypropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-[(1-methylpiperidin-2-yl)methyl]-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
2-[methyl({4-methyl-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol