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(1S,5R)-6-benzyl-3-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-{4-[4-(2-amino-1,3-thiazol-4-yl)phenyl]-1H-pyrazol-1-yl}-N-(2-ethyl-2H-1,2,3-triazol-4-yl)acetamide
5-oxo-1-(propan-2-yl)-N-[2-(pyridin-3-yl)ethyl]pyrrolidine-3-carboxamide
1-ethyl-N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
N-ethyl-1-{[3-(methylsulfanyl)phenyl]methyl}-N-(pyridin-4-ylmethyl)piperidin-3-amine
3-[1-(pyridine-3-sulfonyl)azetidin-3-yl]pyridine
4-{3-[4-(methylsulfanyl)benzoyl]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
(4aR,8aS)-6-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-{[3-(trifluoromethyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
(1R,5R)-6-[(3-chloro-2-fluorophenyl)methyl]-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methyl-4-(4-methylphenyl)piperazine
(5S,9aS,9bS)-5-[2-(furan-2-yl)phenyl]-2-[(2-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-tert-butyl-5-oxo-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)pyrrolidine-3-carboxamide
4-ethyl-5-methyl-6-[4-(1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyrimidin-2-amine
2-(2,5-dimethoxyphenyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
4-{5-[(4-ethyl-2-methyl-3-oxopiperazin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}benzoic acid
5-{1-azabicyclo[3.2.1]octan-5-yloxy}-4-ethyl-7-methyl-2H-chromen-2-one
ethyl (4aS,8aR)-6-(quinoxalin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylate
[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
3-(2-{4-[2-(methylsulfanyl)ethyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
5-(2,6-difluorophenoxymethyl)-N-[3-(1H-indazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
11-({[2-fluoro-5-(trifluoromethyl)phenyl]methyl}amino)-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-[2-(propylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-1H-pyrazole-3-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2,5-dimethylbenzene-1-sulfonamide
methyl 8-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(naphthalen-2-ylmethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-cyclopropyl-1-{1-[(4-fluoro-2-methylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
3-[1-(3-methoxybenzoyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-{3-[({1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}amino)methyl]phenyl}ethan-1-one
methyl (2S,4R)-1-[(2-ethoxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
1-ethyl-5-oxo-N-[(1-phenylcyclohexyl)methyl]pyrrolidine-3-carboxamide
1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-4-(furan-2-carbonyl)-1,4-diazepane
N-(3-methoxypropyl)-1-methyl-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(piperidin-1-yl)piperidine
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-2,5-dihydro-1H-pyrrole-2-carboxamide
(3S)-N,N-dimethyl-1-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]azepan-3-amine
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-2,2-dimethylcyclopropane-1-carboxamide
8-chloro-2-(1,2-oxazolidine-2-carbonyl)quinoline
2-{4-[4-(azepan-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
[2-(4-chlorophenyl)ethyl]({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
2-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-ylmethyl]phenyl}-6-(2-phenylethyl)-3,4-dihydropyrimidin-4-one
[1-({2-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)piperidin-2-yl]methanamine
(1S,5R)-6-cycloheptanecarbonyl-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholine
3-[(3R,4S)-4-(dimethylamino)-1-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}piperidin-3-yl]propanoic acid
5,8-dimethyl-2-({[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]amino}methyl)quinolin-4-ol
5-(2,4-difluorophenoxymethyl)-N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
methyl 3-benzamido-6-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}thieno[2,3-b]pyridine-2-carboxylate
N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-[(3-fluorophenyl)methyl]-4-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]morpholine