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1-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-6-azaspiro[2.5]octane
3-({1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidin-4-yl}oxy)-N-(pyridin-3-ylmethyl)benzamide
7-(1-benzothiophen-3-yl)-4-(1-methyl-1H-pyrazole-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(1H-imidazol-5-yl)-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(1H-pyrrol-1-yl)propanamide
4-hydroxy-2-({3-[(2-methylphenyl)methoxy]azetidin-1-yl}methyl)quinoline-6-carboxamide
5-[1-(1,4-dioxan-2-ylmethyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrazin-2-ol
3-{[(1-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)oxy]methyl}pyridine
5-[1-(5-chloro-2-fluorobenzoyl)piperidin-4-yl]-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
7-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}pyrazolo[1,5-a]pyrimidine-6-carboxamide
5-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-methyl-1H-1,3-benzodiazole
N-[(1-cyclopentylpiperidin-4-yl)methyl]-3-(1,2-oxazolidin-2-yl)-N-(oxolan-2-ylmethyl)propanamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
7-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-cyclohexyl-3-methyl-4-oxo-N-(pyridin-2-ylmethyl)-3,4-dihydroquinazoline-7-carboxamide
2-(methylsulfanyl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyridine-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]ethan-1-one
2-(butylsulfanyl)-6-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
1-[(2-chlorophenyl)methyl]-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
3-({[4-(3-hydroxy-3-methylbutyl)phenyl]formamido}methyl)-N,N-dimethylbenzamide
3-{[1-(4-ethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
1-[(2,6-difluorophenyl)methyl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
N-[4-(4-{[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]amino}piperidin-1-yl)phenyl]pyrazine-2-carboxamide
[1-({4-[(2-chloro-4,5-dimethoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-2-yl]methanol
1-{4-[2-cyclobutyl-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
propan-2-yl 3-{2-[(2-fluorophenyl)carbamoyl]ethyl}piperidine-1-carboxylate
2-methyl-4-(5-{1-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-imidazol-2-yl}thiophen-2-yl)but-3-yn-2-ol
(1R,2S,6R,7S)-4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-azatricyclo[5.2.2.02,6]undecane
2-(4-{[4-(benzyloxy)phenyl]methyl}-1-[(6-methylpyridin-2-yl)methyl]piperazin-2-yl)ethan-1-ol
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-[(5-methyl-1,2-oxazol-3-yl)methyl]urea
5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]-1H-pyrazole-4-carboxamide
3-(3-chlorobenzoyl)-1-cyclobutylpiperidine
N-[(2S,4R,6S)-2-(2-phenylethyl)-6-{2-[(propan-2-yl)amino]pyrimidin-5-yl}oxan-4-yl]acetamide
8-(furan-3-ylmethyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-fluoro-2-methoxybenzamide
N-methyl-N-propyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-4-(2-oxopyrrolidin-1-yl)benzamide
N-(1-ethyl-4-methyl-1H-pyrazol-5-yl)oxane-2-carboxamide
5-methanesulfonamido-N-(oxan-4-ylmethyl)-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-3-yl)-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-cyclopentyl-1-(3-methylbutyl)-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
(3R,4R)-4-cyclobutyl-3-methyl-1-(3-propyl-1H-pyrazole-4-carbonyl)piperidin-4-ol
3-[2-(dimethylamino)ethyl]-8-[(2-fluorophenyl)methyl]-1-[2-(4-methoxyphenyl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-acetamido-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-1-[2-(pyridin-2-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
3-(3-hydroxypyrrolidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
2-[4-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
1-[4-(4-{[2-(3,4-dimethoxyphenyl)ethyl]amino}piperidin-1-yl)benzoyl]piperidin-3-ol
N-[(1-methylpiperidin-4-yl)methyl]-2-(5-oxopyrrolidin-2-yl)-N-(2-phenylethyl)acetamide
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
methyl 6-{2-[(adamantan-1-ylformamido)methyl]-2,3-dihydro-1-benzofuran-7-yl}pyridine-3-carboxylate