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{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
3-{1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-3-carbonyl}pyridine
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-5-(1,2-oxazol-3-yl)thiophene-2-sulfonamide
1-(4-methylpiperazin-1-yl)-3-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-3-yl)propan-1-one
N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-2,3-dihydro-1H-inden-2-amine
5-methyl-N-[(3-methyloxetan-3-yl)methyl]-4-[(3-phenylpropyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-(3-chlorophenyl)-N-[(2S)-3-methylbutan-2-yl]piperidin-4-amine
N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-7-(2-methoxyacetamido)-1-methyl-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
4-{1-[4-(3-chloro-5-methylpyridin-2-yl)phenyl]ethyl}morpholine
4-(4-ethoxy-3-methylphenyl)-N-[(2R)-1-hydroxypropan-2-yl]-4-oxobutanamide
2,6-dimethyl-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}aniline
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-(5-methyl-1,3,4-thiadiazol-2-yl)-10-azabicyclo[4.3.1]decane-10-carboxamide
N-({4-benzyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-(2,5-dimethoxybenzoyl)benzamide
N-{[(2S,4S)-4-fluoro-1-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]pyrrolidin-2-yl]methyl}propanamide
2-(4-acetylphenoxy)-N-[1-(3-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-(2-{7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2,4-dimethylbenzamide
6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-3-(3-fluorophenyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-[(2R,3R)-1'-[(4-acetamidophenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
2-(4-methoxyphenyl)-2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]acetic acid
N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-(3-methylthiophene-2-carbonyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
5-(dimethylamino)-2-(2-oxo-2-{spiro[indene-1,4'-piperidine]-1'-yl}ethyl)-2,3-dihydropyridazin-3-one
N-{[2-(2-ethanesulfonamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(2-fluorophenyl)benzamide
5-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-2-(phenoxymethyl)pyrimidin-4-ol
7-(2,5-dichlorobenzenesulfonyl)-2-methyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-{[4-(trifluoromethyl)phenyl]methyl}benzamide
2-(1-{[3-(carboxymethoxy)phenyl]methyl}pyrrolidin-3-yl)benzoic acid
1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[(3,5-dimethylphenyl)methyl]-4-(2-methoxybutanoyl)piperazin-2-one
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-5-hydroxy-N-methylpyrazine-2-carboxamide
5-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1H-1,2,4-triazol-3-amine
4-(quinoxalin-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-amino-2-methyl-N-[1-(4-phenylphenyl)ethyl]propanamide
diphenyl({1-[(2R)-pyrrolidine-2-carbonyl]piperidin-4-yl})methanol
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
2-[(3-carbamoylpiperidin-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(3S,4R)-1-(3-phenyl-1,2-oxazole-4-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-(1H-imidazol-4-yl)-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]acetamide
3-chloro-N-(2-methoxyethyl)-4-[(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)oxy]benzamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(1,3-thiazole-4-carbonyl)piperazin-2-yl}ethan-1-ol
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
2-(morpholin-4-yl)-1-[(3S,4R)-3-(propan-2-yl)-4-[(1,3-thiazol-2-yl)amino]pyrrolidin-1-yl]ethan-1-one
3-({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)-3-methyl-1λ6-thiolane-1,1-dione
1-[3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)propanoyl]piperidine-3-carboxylic acid
2-{2-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
(4aS,8aR)-6-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine