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3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]benzamide
{7-fluoro-5-[6-(piperidine-1-carbonyl)pyrazin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
N-propyl-4-{[3-(1H-pyrazol-1-yl)propyl]amino}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
N-cyclopropyl-1-[1-(2-hydroxyacetyl)piperidin-4-yl]piperidine-3-carboxamide
2-(methylsulfanyl)-5-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-3,4-dihydropyrimidin-4-one
N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-2,3-dihydro-1H-indene-1-carboxamide
5-(1-methylpyrrolidin-3-yl)-3-(3-phenylpropyl)-1,2,4-oxadiazole
N-(2-cyclopentyl-2-phenylethyl)-3-(1,2-oxazinan-2-yl)propanamide
1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-[2-(dimethylamino)ethyl]-N-(2-hydroxyethyl)-6-oxo-N-(1,3-thiazol-2-ylmethyl)piperidine-3-carboxamide
N-{2-[(4-chlorophenyl)methoxy]ethyl}-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
(3S,9R)-11-(4-methylbenzoyl)-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
1-{2-oxo-2-[6-oxo-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}imidazolidine-2,4-dione
2-{[(3S)-3-aminopiperidin-1-yl]methyl}-6-fluoroquinolin-4-ol
(2R,6R)-11-methoxy-4-[(4-methyl-1H-imidazol-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N,5-dimethyl-N-(2-phenylethyl)-4-[(pyridin-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-(3-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-oxopropyl)azepan-2-one
N-({8-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
5-(methoxymethyl)-N-{3-methyl-1-[7-(3-methylbutyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]butyl}furan-2-carboxamide
N-cyclohexyl-3-(1-methyl-1H-pyrazol-4-yl)-N-(thiophen-3-ylmethyl)propanamide
6-cyano-N-[(3R,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]pyridine-3-carboxamide
4-[(2-methylprop-2-en-1-yl)oxy]-N-[2-(methylsulfamoyl)ethyl]benzamide
N-benzyl-3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
N-butyl-N-[(4-fluorophenyl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
5,6-dimethyl-2-oxo-N-[1-(thiophen-3-yl)propan-2-yl]-1,2-dihydropyridine-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methylpropanamide
8-(2-{[(4-fluorophenyl)methyl](methyl)amino}acetyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
2-[1-(2-hydroxyethyl)-5-(2,3,4-trimethoxyphenyl)-1H-1,2,4-triazol-3-yl]acetamide
8-chloro-2-{1-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1H-imidazol-2-yl}quinoline
2-{[4-(2-chlorophenyl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
1-cyclohexyl-3-(2-methoxyethyl)-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
N-(3-chloro-4-methoxyphenyl)-6-[(2E)-3-(2,3-difluorophenyl)prop-2-enoyl]-6-azaspiro[2.5]octane-1-carboxamide
4-{[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
1-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-3-(1-methyl-4-phenyl-1H-pyrazol-5-yl)urea
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1-methyl-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}urea
6-[(3-fluorophenyl)methoxy]-1-(2-methylpropyl)-4-(4,4,4-trifluorobutanoyl)-1,4-diazepan-2-one
N-[(5-chlorothiophen-2-yl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-ethyl-7-(2-methoxybenzamido)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
methyl (2S,3S)-3-methyl-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)pentanoate
2-{2-chloro-4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]phenoxy}acetamide
4-(1-methyl-1H-imidazol-2-yl)-1-[(2,3,6-trifluorophenyl)methyl]piperidine
methyl 3-cyclohexaneamido-5-{[(1-methyl-1H-pyrazol-5-yl)formamido]methyl}benzoate
3-(1,2-diethyl-1H-1,3-benzodiazol-5-yl)-1-[(4,6-dimethylpyridin-3-yl)methyl]urea
4-{[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-methyl-1H-pyrazole
(2S,4R)-1-[(3,4-difluorophenyl)methyl]-N-[2-(dimethylamino)ethyl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
methyl 8-(2,3-difluorobenzoyl)-1-(2-methoxyethoxy)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-N-methyl-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
5-methyl-1-{3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}-1H-1,2,3,4-tetrazole
5-[4-(aminomethyl)piperidin-1-yl]-2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2,3-dihydropyridazin-3-one
N-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide