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({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-(furan-2-ylmethyl)-5-methylthieno[2,3-d]pyrimidin-4-amine
3-(2-fluorophenyl)-5-(4-methoxybenzenesulfonyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
N-(2-ethyl-2H-1,2,3-triazol-4-yl)-2-[5-(3-hydroxyphenyl)-1H-indazol-1-yl]acetamide
5-methyl-1-(4-{4-[(3-methylbutan-2-yl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
4-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methylphenol
N'-[2-(azepan-1-yl)ethyl]-N-(2,4-dimethylphenyl)-N'-methylpropanediamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(4-fluorophenyl)-1,4-diazepane
4-(hydroxymethyl)-1-[3-(2-methoxyphenoxy)propyl]azepan-4-ol
N-(1-{7-[(4-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-(1,3-benzothiazol-2-yl)-1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]propan-1-one
N-(1-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
6-cyclopentyl-3-[1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl]-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(3-methylphenyl)pyridine-3-carboxylic acid
methyl 8-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indazole
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxybenzoyl)piperidine
1-benzyl-N-cyclopropyl-4-oxo-5-(4-phenyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-methyl-3-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]imidazo[1,2-a]pyridine
8-[(4-fluoro-3-methoxyphenyl)methyl]-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-2-(4-phenylphenyl)ethan-1-one
2-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-4H-chromen-4-one
N-[4-(1H-indol-2-yl)phenyl]-1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidine-4-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-4-phenyl-N-(pyridin-2-ylmethyl)benzamide
(3S,4R)-4-(3-fluorophenyl)-1-[3-(methylsulfanyl)propyl]pyrrolidine-3-carboxylic acid
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]urea
2-{4-[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]piperazin-1-yl}ethan-1-ol
6-chloro-2-{1-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-(2-chloro-4-fluorophenyl)-N-({5-methyl-2-[2-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)acetamide
5-(2-{[(3-fluorophenyl)methyl]amino}ethyl)-1-[2-(propan-2-yloxy)ethyl]pyrrolidin-2-one
2-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}benzoic acid
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]acetamide
N-(oxolan-2-ylmethyl)-2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(3-chlorophenyl)-4-{1-[(2E)-4-methylpent-2-en-1-yl]piperidin-3-yl}piperazine
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
4-({6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)-5-cyclopropyl-1-methyl-1H-pyrazole
4-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)pyridine
5-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
methyl 1-(2-methoxyethoxy)-2-oxo-8-(2,5,7-trimethylquinoline-4-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylate
5-{[4-(adamantan-1-yl)piperazin-1-yl]methyl}-2-propylpyrimidine
2-(dimethylamino)-N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methylpyrimidine-5-carboxamide
2-[2,5-dioxo-3-phenyl-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}acetamide
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
[(3R,4R)-1-[3-(dimethylamino)pyrazin-2-yl]-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(2H-1,3-benzodioxol-5-yl)-5-(3,4,5-trimethoxyphenoxymethyl)-1,2,4-oxadiazole
methyl({[3-({1-[4-(morpholin-4-yl)benzoyl]piperidin-4-yl}oxy)phenyl]methyl})(2-phenylethyl)amine
7-fluoro-3-{[(2-hydroxy-2-phenylethyl)(methyl)amino]methyl}-1-(pyridin-4-ylmethyl)-1,2-dihydroquinolin-2-one
4-methyl-6-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyrimidin-2-amine