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2-methoxy-4-[(1E)-3-[3-(pyrrolidin-1-yl)piperidin-1-yl]prop-1-en-1-yl]phenol
(4aS,8aR)-1-(2-aminoethyl)-6-({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-decahydro-1,6-naphthyridin-2-one
(3aR,6aR)-2-cyclopentyl-N-[2-(4-hydroxy-1-methylpiperidin-4-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-methyl-3-(3-methylpiperidin-1-yl)-N-[2-(piperidin-1-yl)ethyl]propanamide
11-{[(2,6-difluorophenyl)methyl]amino}-4-(quinolin-3-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-ethyl-N-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
3-[4-(2-methylpropyl)-1H-pyrazol-5-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidine
[1-(3-chlorobenzoyl)-4-[(3-methoxyphenyl)methyl]piperidin-4-yl]methanol
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylbutanamide
1-methyl-5-{[2-(methylsulfanyl)ethyl]amino}-N-(thiophen-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-(1-{7-[(2,4,6-trimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)pyridine-3-carboxamide
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
3-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}benzoic acid
(2S,4R)-4-(5-chloro-2-fluorobenzamido)-1-(1H-imidazol-4-ylmethyl)-N-methylpyrrolidine-2-carboxamide
(3aS,6aS)-2-(2,3-dihydro-1H-inden-2-yl)-5-(ethanesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-hydroxyethan-1-one
(4aR,7aS)-N,N-dimethyl-4-[(2-methylpyrimidin-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
ethyl 1-[(5-ethylthiophen-2-yl)sulfonyl]-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
2-benzyl-4-[(E)-2-(furan-2-yl)ethenyl]-3-methyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(3R,4R)-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-3,4-dimethylpyrrolidin-3-ol
2-amino-6-(1,2-dimethyl-1H-indol-3-yl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-3-(4-methoxyphenyl)-1-(3-methylbutyl)pyrrolidine-2,5-dione
(2S,4S)-4-[4-({[(4-fluorophenyl)carbamoyl](methyl)amino}methyl)-1H-1,2,3-triazol-1-yl]-N-methylpyrrolidine-2-carboxamide
3-[3-({[(1-ethylpyrrolidin-2-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
4-[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]-5-ethyl-2-methylpyrimidine
3-ethyl-1-(2-phenylethyl)-8-{[4-(trifluoromethoxy)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
methyl 9-(benzyloxy)-3-[(2,4-dimethoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
6-[(5-acetylthiophen-3-yl)methyl]-2-(2-hydroxyethyl)-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
methyl 3-(2-methylpropyl)-2-oxo-1-(1,3-thiazol-2-ylmethyl)-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
methyl 4-{[(2-{1-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-5-oxopyrrolidin-2-yl}ethyl)amino]methyl}benzoate
N-benzyl-N-ethyl-3-{5-[methoxy(phenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
1-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-4-(hydroxymethyl)piperidin-4-ol
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-3-carboxamide
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-[(4-fluorophenyl)methyl]-3-(2-phenylacetyl)piperidine-1-carboxamide
N4-cyclobutyl-7-[(4-methyl-1,3-thiazol-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-(2-methylphenyl)-4-[4-(propan-2-yl)benzoyl]piperazin-2-one
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-1-(methoxymethyl)cyclobutane-1-carboxamide
(3aS,6aS)-2-methyl-5-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-(2-methylphenyl)-4H-1,2,4-triazol-3-yl)methyl]-2-methyl-1,3-thiazole-4-carboxamide
1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-2-(pyridin-3-yl)ethan-1-one
1-(azocan-1-yl)-3-(4-{[(dicyclopropylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}-4-{[4-(methylsulfanyl)phenyl]methyl}piperazine
N-[(1-methylpiperidin-4-yl)methyl]-5-[(methylsulfanyl)methyl]-N-(2-phenylethyl)furan-2-carboxamide
1-{1-[5-(1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]butan-2-yl}-4-methylpiperazine
methyl (2S,4R)-1-[(3-ethoxy-4-methoxyphenyl)methyl]-4-{2-[4-(trifluoromethyl)phenyl]benzamido}pyrrolidine-2-carboxylate
N-butyl-1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
4-chloro-3-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1-methyl-1H-indazole