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N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)furan-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(pyridin-4-ylmethyl)piperidin-3-yl]piperazine
3-{5-[2-(pyridin-4-yl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2,4,5-trifluoro-N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)benzamide
N-{1-[(4-fluorophenyl)methyl]-5-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1H-1,3-benzodiazol-7-yl}acetamide
1-[(4-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)pyridine-3-carbonyl]-6-(pyridin-4-ylmethoxy)-1,4-diazepan-2-one
2-(ethylamino)-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methyl-1,3-thiazole-5-carboxamide
ethyl 4-{[(4-methylphenyl)(pyridin-4-yl)methyl]amino}piperidine-1-carboxylate
1-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(1H-imidazol-1-ylmethyl)-1-[4-(piperidin-1-ylmethyl)benzoyl]piperidine
1-[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
2-(3-methylbutyl)-8-(1,3-thiazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(3-fluorophenyl)piperazin-2-one
2-(3-methoxyphenyl)-3-[(3-methoxypiperidin-1-yl)methyl]-7-(methylsulfanyl)quinoline
1-(3-methoxybenzoyl)-4-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
4-(2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-oxoethyl)-5-methyl-2,3-dihydro-1H-pyrazol-3-one
2-(pyridin-2-ylsulfanyl)-N-{[7-(pyrimidin-2-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}acetamide
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-{6-oxa-9-azaspiro[4.5]decan-9-yl}ethan-1-one
1-{4-[4-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]phenyl}ethan-1-one
[(3R,4R)-1-[1-(4-chlorophenyl)cyclohexanecarbonyl]-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-2,2-diphenyl-N-(pyridin-4-ylmethyl)acetamide
4-({2-[3-(dimethylamino)propoxy]phenyl}methyl)-N,N-dimethylpiperazine-1-carboxamide
8-(2,3-dimethylquinoxaline-6-carbonyl)-1-[(2-fluorophenyl)methoxy]-1,8-diazaspiro[4.5]decan-2-one
2-cyclopropyl-9-(2,2-dimethylpropanoyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
[2-(1H-1,3-benzodiazol-2-yl)ethyl][1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
N-(2-{1-[1-(diphenylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}ethyl)acetamide
1-[4-(4-acetylphenyl)piperazin-1-yl]-3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
5-[2-(methylamino)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
2-[(furan-3-ylmethyl)(methyl)amino]-2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}acetic acid
N-({2-[2-(2-cyclopentylacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-3,5,7-trimethyl-1H-indole-2-carboxamide
4-ethyl-3-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[2-methyl-3-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)-1H-indol-1-yl]acetamide
3-ethyl-1-(5-fluoro-2-methoxyphenyl)-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
4-chloro-3-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}-N-methylbenzamide
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]acetamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[(2-methylphenyl)(pyridin-4-yl)methyl]amine
1-(3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carbonyl)piperidine
1-(furan-2-ylmethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylic acid
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-1-benzothiophene-2-carboxamide
5-[6-(morpholin-4-yl)pyrimidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,4-diazepan-5-one
1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-methyl-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
4-[1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}phenyl)ethyl]morpholine
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]benzamide
2-(dimethylamino)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-(4-methylphenyl)acetamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-5-(naphthalen-2-yl)-1,2,4-triazin-3-amine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(oxolan-3-yl)-1,2-oxazole-3-carboxamide
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenylpropanamide
1-[1-(2-fluoro-6-methoxybenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol