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4-{6-[4-(piperidin-1-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
1-(1H-pyrazole-4-carbonyl)-3-(trifluoromethyl)piperidine
1-[3-methoxy-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)phenyl]-1H-1,2,3,4-tetrazole
N-({7-[2-(cyclohex-1-en-1-yl)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyridin-3-yl)propanamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-(prop-2-en-1-yl)-1,2,4-oxadiazole
1-{3-[5-(3-fluoro-5-methylphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
N-cyclopropyl-2-ethyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}butanamide
2-(dimethylamino)-N-(3-{[(furan-2-ylmethyl)(2-hydroxyethyl)carbamoyl]amino}-2-methylphenyl)acetamide
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]-5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-4-(5-methyl-1,3,4-oxadiazol-2-yl)-1,4-diazepane
3-benzyl-8-[(3-hydroxy-4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-(1,3-thiazol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-ethyl-8-methyl-2-[2-(methylamino)pyrimidin-5-yl]-N-(pyridin-2-ylmethyl)quinoline-4-carboxamide
[3-(3-methylbut-2-en-1-yl)-1-(1H-pyrazole-3-carbonyl)piperidin-3-yl]methanol
N-methyl-4-(1H-pyrazol-4-yl)-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}butanamide
5-(5-chloro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-2-methyl-1,4-dihydropyridin-4-one
2-[4-(2H-1,3-benzodioxol-4-ylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
4-[4-({4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
ethyl 4-(4-{4-[(3-ethoxypropyl)amino]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
5-cyclopropyl-N-[2-(diethylamino)ethyl]-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)pent-4-enamide
4-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]-1λ6-thiomorpholine-1,1-dione
5-acetyl-N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentylthiophene-3-carboxamide
8-(5-propylpyrimidin-4-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]-N-(pyrimidin-4-ylmethyl)acetamide
2-methyl-N-({8-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-thiazole-4-carboxamide
N-benzyl-N-(cyclopropylmethyl)-2-[1-ethyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
5-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]quinoxaline
N-(1-{7-[(3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-phenoxyacetamide
3-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-1-[2-(morpholin-4-ylmethyl)phenyl]urea
(3S,4S)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
1-cyclohexyl-3-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-3-(2-fluorophenyl)pyrrolidine-2,5-dione
4-[1-(3,4,5-trimethoxyphenyl)-1H-imidazol-2-yl]-2,1,3-benzoxadiazole
2-[4-(ethylamino)pyrimidin-2-yl]-N,N-bis(propan-2-yl)benzamide
N-(4-{[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]methyl}phenyl)acetamide
3-{1-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]piperidin-4-yl}-N-[(3-chlorophenyl)methyl]propanamide
1-[(2S,4R)-1-[(2,4-dimethylphenyl)methyl]-4-[(4,6-dimethylpyrimidin-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
(3R,9aR)-3-[(1S)-1-hydroxyethyl]-8-[4-(trifluoromethoxy)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-2-(morpholin-4-yl)-N-[2-(pyridin-3-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
5-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[3-(4-chloro-1H-pyrazol-1-yl)propyl]-3-(3-ethyl-1,4-dimethyl-1H-pyrazol-5-yl)urea
1-[(5-{[4-(difluoromethoxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]-3,3-dimethylurea
3-chloro-N-cyclopentyl-4-({1-[4-(methylsulfanyl)butan-2-yl]piperidin-4-yl}oxy)benzamide
(3aR,6aS)-2-[(2,4-difluoro-3-methoxyphenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole
5-methyl-N-{2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
1-phenyl-N-({1-[2-(thiophen-3-yl)acetyl]piperidin-3-yl}methyl)methanesulfonamide
6-chloro-3-{[7-(1-hydroxy-2-phenylethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-4H-chromen-4-one
1-[9-hydroxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yloxy)ethan-1-one