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2-(1H-1,3-benzodiazol-1-ylmethyl)-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1,3-oxazole-4-carboxamide
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(1,2-oxazol-5-ylmethyl)acetamide
2-{1-[(4-fluorophenyl)methyl]-4-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(1-{7-[(2,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
1-(oxolane-2-carbonyl)-4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]piperidine
4-(2-fluorophenyl)-2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-(propan-2-yl)-1H-pyrazol-1-yl}pyrimidine
5-(4-fluorophenyl)-3-[2-(4-fluorophenyl)pyrrolidin-1-yl]-1,2,4-triazine
N-(2-methoxyethyl)-5-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(diphenylmethyl)-N-{2-[(2R)-pyrrolidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
N-{[8-(thiophene-2-sulfonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-(2,4,6-trifluorophenyl)acetamide
1-(2-{6-[(3-fluorophenyl)methoxy]-4-(2-methylpropyl)-3-oxo-1,4-diazepane-1-carbonyl}phenyl)-1,3-diazinane-2,4-dione
3-(5-fluoro-2-methoxybenzoyl)-1-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidine
6-(3-fluoro-4-methoxybenzoyl)-N-[2-(3-methoxyphenyl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
5-[(3-fluorophenyl)methyl]-5-{1-[(2E)-3-(4-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
N-(2,3-dihydro-1-benzofuran-3-yl)-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
N-cyclopentyl-2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)acetamide
(2S,4R)-1-cycloheptyl-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
ethyl 4-{1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl}piperazine-1-carboxylate
2-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]ethan-1-one
N-(3,5-dimethylphenyl)-6-(3-phenylprop-2-ynoyl)-6-azaspiro[2.5]octane-1-carboxamide
1-[(2-fluorophenyl)methyl]-6-oxo-N-[3-(1H-pyrazol-1-yl)propyl]piperidine-3-carboxamide
1-methyl-4-{[(3S,5R)-1-(2-phenylethyl)-5-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}piperazine
{1-[1-(2,3-dihydro-1-benzofuran-5-ylmethyl)piperidin-4-yl]-2-phenylethyl}(2-methoxyethyl)(pyridin-3-ylmethyl)amine
N-[(2-ethoxypyridin-3-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
2-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-3,4-dihydroquinazolin-4-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
methyl 4-(5-{[(1-benzothiophen-2-ylmethyl)(methyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
1-(furan-2-ylmethyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}propanamide
4-(1-butyl-1H-imidazol-2-yl)-N-(4-methoxyphenyl)piperidine-1-carboxamide
4-(1-benzofuran-2-carbonyl)-6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
5-(2,3-dihydro-1H-inden-2-yl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
3-[1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
N-ethyl-N-{2-phenyl-1-[1-(quinolin-4-ylmethyl)piperidin-4-yl]ethyl}oxane-4-carboxamide
7-(6,7-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-cyclopentanecarbonyl-N-[(5-methylpyrazin-2-yl)methyl]piperidine-4-carboxamide
N-[2-(4-{[2-(3,4-dimethoxyphenyl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-3-carboxamide
5,6-dimethyl-2-oxo-N-[(2,3,4-trifluorophenyl)methyl]-1,2-dihydropyridine-3-carboxamide
1-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 2-[(4-hydroxyquinolin-2-yl)methyl]-2,7-diazaspiro[4.5]decane-7-carboxylate
N-(5-fluoropyridin-3-yl)-3-[(oxolan-3-ylmethyl)sulfamoyl]benzamide
2-amino-N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-methyl-1,3-benzothiazole-6-carboxamide
3-(4-hydroxyphenyl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-pyrazole-5-carboxamide
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-3-sulfamoylthiophene-2-carboxamide
N-(3,4-dimethylphenyl)-3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
5-{1-[2-(2,3-difluorophenyl)acetyl]piperidin-4-yl}-3-[2-(4-methoxyphenyl)ethyl]-5-methylimidazolidine-2,4-dione
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-[2-(pyridin-4-ylsulfanyl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl]methanol
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3S,4R)-3-(dimethylamino)-N-(furan-2-ylmethyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide