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3-[2-(dimethylamino)ethyl]-5-[(3-fluorophenyl)methyl]-5-[1-(1-methylcyclohexanecarbonyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(2-hydroxyethyl)-2,4-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidine-5-carboxamide
1-[2-(morpholin-4-yl)ethyl]-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
3-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-[3-({[(2-chlorophenyl)methyl](2-hydroxyethyl)carbamoyl}methoxy)phenyl]propanamide
2-[8-(1-methyl-1H-pyrrole-2-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
3-(2,3-dihydro-1H-inden-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[(4aR,7aS)-4-[(4-fluoro-3-methoxyphenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]-1,3-thiazole-4-carboxamide
1-benzyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
8-chloro-N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]quinoline-2-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
1-(2-methylpropyl)-4-[(2S)-5-oxopyrrolidine-2-carbonyl]-6-(pyridin-3-ylmethoxy)-1,4-diazepan-2-one
methyl 2-[(1-methoxypropan-2-yl)sulfamoyl]-6-(3-phenylpropyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-methyl-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-phenylpiperidine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
N3-(adamantan-1-ylmethyl)-1-(butan-2-yl)-N5-ethyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3Z)-hex-3-en-1-yl]-7-hydroxy-6-methyl-1,2,3,4-tetrahydroquinolin-2-one
3-[(3-fluorophenyl)methyl]-N-[2-(propan-2-yloxy)ethyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-4,6-dimethylpyrimidine
(3aR,6aR)-2-acetyl-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[2-methyl-1-(morpholin-4-yl)propan-2-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
5-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-[2-(1H-imidazol-1-yl)ethyl]-4-phenyl-1H-imidazole
N-methyl-2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[(1-methylpyrrolidin-3-yl)methyl]-1,3-oxazole-4-carboxamide
(3R,4R)-3-cyclobutyl-1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-methylpyrrolidin-3-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
5-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
(5S,9aS,9bS)-2-phenyl-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(6-methylpyridin-2-yl)piperazine
4-(1-{imidazo[1,2-a]pyridine-2-carbonyl}pyrrolidin-3-yl)-1-(2-methylpropyl)piperidine
5-methyl-1'-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N'-(3-chloro-2-methylphenyl)-N-[1-(1H-1,2,4-triazol-5-yl)ethyl]propanediamide
[(3-cyclohexyl-1H-pyrazol-4-yl)methyl](methyl)[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amine
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)[(3-methyl-1,2-oxazol-5-yl)methyl]amine
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-methylpyrazine-2-carboxamide
5-({[(3-{2-[4-(5-chloro-2-methoxybenzenesulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)amino}methyl)pyrrolidin-2-one
3-{[(4,6-dimethylpyrimidin-2-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
N3-(3-methylbutyl)-1-(2-methylpropyl)-4-oxo-N5-[3-(pyridin-4-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-3-(2-methylphenyl)propan-1-one
3-(2,3-dihydro-1H-inden-5-yl)-1-{[4-(dimethylamino)oxan-4-yl]methyl}urea
7,7-dimethyl-2-(1,3-thiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}ethan-1-one
2-tert-butyl-6-(2,6-difluoro-3-methylbenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-methylimidazo[1,2-a]pyrimidine-3-carboxamide
N3-[(2,3-dimethyl-1H-indol-5-yl)methyl]piperidine-1,3-dicarboxamide
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-ethyl-2-methyl-1,3-thiazole-5-carboxamide
5-[2-(2-phenylethyl)morpholine-4-carbonyl]-1H-1,2,3-benzotriazole