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N-methyl-3-(piperidin-3-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
(1S,4S)-2-(2-chlorophenyl)-5-[(4-methoxy-2,3-dimethylphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
4-{9-methoxy-3-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}piperazin-2-one
2-cyclopropyl-9-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
N-[3-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
methyl 8-{[2-(difluoromethoxy)phenyl]methyl}-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-{[(4-fluorophenyl)methyl]amino}-N-[3-(morpholin-4-yl)propyl]benzamide
4-(cyclopropylmethyl)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
5-{[benzyl(methyl)amino]methyl}-N-[2-(furan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]propanamide
ethyl 1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
4-(1-cyclopentyl-6-oxopiperidine-3-carbonyl)-1-(3,5-dimethylphenyl)piperazin-2-one
N-cyclohexyl-3-(4-hydroxyphenyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-5-carboxamide
3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}-1-(propan-2-yl)piperidine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-[(2-methylphenyl)methyl]piperazine
5-[(6,7-dimethoxy-4-methylquinolin-2-yl)amino]pentan-1-ol
6-[(3-ethoxy-4-hydroxyphenyl)methyl]-N-{[3-(trifluoromethyl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
6-[4-(pyrrolidin-3-yl)piperidin-1-yl]pyridine-3-carboxamide
2-methyl-4-oxo-N-(2,4,4-trimethylpentan-2-yl)-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
1-(benzenesulfonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(3S,5S)-1-(3-methoxypropanoyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
1-{4-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]phenyl}pyrrolidin-2-one
2-(dimethylamino)-2-(2-methylphenyl)-N-[3-oxo-3-(pyrrolidin-1-yl)propyl]acetamide
3-{[2-(5-methylfuran-2-yl)ethyl]sulfamoyl}-N-(pyrrolidin-3-yl)benzamide
3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
1-methyl-N-({8-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1H-pyrazole-3-carboxamide
1-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]isoquinoline
8-[(2,3,4-trifluorophenyl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
3-({1-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]propan-2-yl}oxy)pyridine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(morpholin-4-yl)benzamide
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-{[4-(1H-pyrazol-1-yl)butan-2-yl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-methyl-1-[(3-methylphenyl)methyl]-4-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazin-2-one
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-5-cyclopropyl-1,3-oxazole-4-carboxamide
5-(2-methoxy-2-phenylacetyl)-1-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
1-ethyl-3-{2-[4-(1-hydroxypropyl)piperidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
1-(3-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
3-(1-{1-[2-(2-fluorophenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-N-(pyridin-4-ylmethyl)cyclohexanecarboxamide
2-(dimethylamino)-2-(4-methylphenyl)-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]ethan-1-one
N,N-dimethyl-2-(4-{5-[(1E)-prop-1-en-1-yl]-2-(pyridin-3-yl)pyrimidin-4-yl}piperidine-1-carbonyl)aniline
N-[1-(furan-2-yl)ethyl]-9-methoxy-3-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{2-[(4-benzyl-5-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}morpholine
1-[4-(4-methyl-1H-pyrazol-3-yl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
6-(4-hydroxypiperidin-1-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
2-[(6-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}pyrimidin-4-yl)amino]ethan-1-ol
N-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
6-[4-(adamantan-2-yl)piperazin-1-yl]-N-(3-methoxypropyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-{1-[(4-fluorophenyl)methyl]-1H-pyrazol-3-yl}-4-methyl-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,3-thiazol-2-amine