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N-[(4,6-dimethylpyrimidin-2-yl)methyl]-1-(6-ethoxy-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
3-(pyrrolidin-1-yl)-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-(morpholin-4-yl)ethan-1-one
6-fluoro-2-{[4-(thiomorpholin-4-yl)piperidin-1-yl]methyl}quinolin-4-ol
(2R,6R)-1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-{2-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[(4-phenyl-1,3-thiazol-5-yl)methyl]propanamide
N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[1-(3-chlorobenzoyl)piperidin-4-yl]-5-(2-methylphenyl)-2-(pyridin-3-yl)pyrimidine
3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(4-methoxyphenyl)-6,6-dimethyl-4-[3-(1H-pyrazol-1-yl)benzoyl]piperazin-2-one
2-[2-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-2-oxoethyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(6-methylpyridin-2-yl)methyl]propanamide
(1S,5R)-6-[(2,3-difluoro-4-methylphenyl)methyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
methyl 6-[2-(2-fluorophenyl)acetyl]-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-2-phenylethan-1-ol
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetamide
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}pyridine-3-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-2,3-dimethyl-1H-indole-7-carboxamide
5-methyl-N-[(1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]-1,2-oxazole-3-carboxamide
2-(4-methoxyphenyl)-3-[(3-methoxypiperidin-1-yl)methyl]-7-methylquinoline
2-[4-(2-ethylpiperidine-1-carbonyl)-5-(methoxymethyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
4-chloro-1-methyl-3-{[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]methyl}-1H-indazole
4-methyl-2-propyl-5-[(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
4,6-dimethyl-2-oxo-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
2-methoxy-4-[4-(1-methoxyethyl)phenyl]pyridine-3-carbonitrile
3-butanamido-N-[2-(4-ethyl-1,3-thiazol-2-yl)ethyl]benzamide
5-(2-chloro-4-fluorobenzoyl)-N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(3S,4R)-1-[(5-methylthiophen-2-yl)methyl]-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})(pyridin-4-ylmethyl)amine
[1-(1,2-oxazol-3-ylmethyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
methyl 6-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylate
N-(1,3,4-thiadiazol-2-yl)-10-azabicyclo[4.3.1]decane-10-carboxamide
(4-{[1-(4-methylpiperidine-4-carbonyl)pyrrolidin-3-yl]methyl}phenyl)methanol
2-methyl-4-(4-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}phenyl)butan-2-ol
1-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-4-(1H-pyrazol-1-yl)butan-1-one
(1S,5R)-3-{2-[4-(hydroxymethyl)phenyl]acetyl}-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-{5-[(3-benzoylpiperidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}pyridine
[(2-ethoxyphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
1-(2-methylphenyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-1,4-diazepane
1-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-4-phenylpiperidine
methyl 4-(4-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)benzoate
N-[2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
1-(2-chlorophenyl)-4-{[2-(2-hydroxyethoxy)phenyl]methyl}piperazin-2-one
3-[(3S,4R)-1-[(2,3-dimethoxyphenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-[(3-fluorophenyl)methyl]propanamide
ethyl({[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
[(4-fluoro-3-methylphenyl)methyl](methyl)[3-(1H-pyrazol-1-yl)propyl]amine