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N-(3-hydroxyadamantan-1-yl)pyrazolo[1,5-a]pyridine-7-carboxamide
N-[3-(cyclopentyloxy)phenyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
N-[(2,4-difluorophenyl)methyl]-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]acetamide
N'-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)ethanediamide
N-[(2-methoxyphenyl)methyl]-1-[4-methyl-6-(propan-2-yl)quinazolin-2-yl]piperidine-4-carboxamide
N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-2,3-dihydro-1,4-benzodioxine-6-carboxamide
6-(1-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}piperidin-4-yl)-2-methylpyrimidin-4-ol
1-methyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(pyridin-3-yl)propyl]acetamide
(1-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}piperidin-2-yl)methanamine
ethyl 4-{6-[(2,3-dimethoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
1-(2,3-dihydro-1H-inden-2-yl)-4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
(3S,4S)-N-(2,3-difluorophenyl)-3-hydroxy-4-(piperidin-1-yl)pyrrolidine-1-carboxamide
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
3-[2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]-1,3-oxazinan-2-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-methyl-1-[(methylcarbamoyl)methyl]-1H-pyrazole-3-carboxamide
5-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-5-[(4-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-[3-(4-methoxy-2-methylphenyl)benzoyl]-1-methyl-1H-imidazole
3-[7-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
1-{4-[(4-acetylphenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methylthiophen-2-yl)methyl]piperidine
ethyl 2-(4-{1-[(2-chloro-4-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}morpholin-3-yl)acetate
(2S,4R)-4-amino-N-ethyl-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidine-2-carboxamide
methyl 3-[(1-cyclopentyl-6-oxopiperidin-3-yl)formamido]propanoate
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2-fluorophenyl)methyl]-N-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-4-(2-phenoxyethyl)piperazine
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2,3,4-trimethoxy-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)benzamide
3-[1-(3,6-dimethyl-1-benzofuran-2-yl)-N-(2-phenylethyl)formamido]propanamide
1-(4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}thiophen-2-yl)ethan-1-one
3-[1-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)piperidin-3-yl]benzoic acid
4-{2-[(4-chlorophenyl)methyl]benzoyl}-2-(trifluoromethyl)morpholine
[(2,3-difluorophenyl)methyl](ethyl){[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
1-(cyclopropylmethyl)-5-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(3,5-dimethoxyphenyl)-5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridine
2-chloro-4-(1-propyl-1H-1,2,4-triazol-5-yl)benzamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N3-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}piperidine-1,3-dicarboxamide
6-(methoxymethyl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyrimidin-4-amine
N-[2-(2-chlorophenyl)-2-hydroxyethyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
3-(cyclopropylmethyl)-5-[(4-fluorophenyl)methyl]-5-[1-(furan-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-1,2,4-triazol-3-yl]pyridine
N-[2-(4-fluorophenyl)ethyl]-N-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}cyclobutanecarboxamide
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-[2-(pyridin-2-yl)ethyl]acetamide
2-{[5-({3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)furan-2-yl]sulfanyl}pyrimidine
5-[(diethylcarbamoyl)methyl]-N-[(4-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[2-({3-methyl-3,9-diazaspiro[5.6]dodecan-9-yl}methyl)phenoxy]acetic acid