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methyl 5-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
4-(3-ethenylphenyl)-5,7-dimethoxy-1,2,3,4-tetrahydroquinolin-2-one
2-(2-methoxyethyl)-6-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1,3-benzoxazole
2-ethyl-7-methoxy-4-[(3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-ethyl-1-{4-[3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}butan-1-one
2-[2-(dimethylamino)ethyl]-9-(2-methyl-3-phenylcycloprop-2-ene-1-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(1H-imidazol-1-yl)propyl]benzamide
N-{2-[4-(dimethylamino)phenyl]ethyl}-5-methyl-1,3-oxazole-4-carboxamide
4-{[(2S,4S)-2-[4-(2-fluorophenyl)piperazine-1-carbonyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidin-1-yl]methyl}-2-methoxyphenol
3-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-N-(1,2,3-thiadiazol-5-yl)benzamide
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-[2-(4-phenylphenyl)acetyl]-1,4-diazepan-5-one
3-phenoxy-N-{1-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}propanamide
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}piperidin-4-amine
2-ethyl-7-(2-methoxybenzamido)-1-methyl-N,N-bis(prop-2-en-1-yl)-1H-1,3-benzodiazole-5-carboxamide
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-(2-{7-[2-(4-chlorophenoxy)acetyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-2-methylpropanamide
3-(3-benzoylpiperidin-1-yl)-5-(1-benzofuran-2-yl)-1,2,4-triazine
N-(propan-2-yl)-1-{2-[1-(pyridin-2-ylmethyl)piperidin-2-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
1-[4-(2-phenoxyethyl)piperazin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-4-yl)thiomorpholine
3-(6-cyanopyridin-3-yl)-1-methyl-1-(thian-4-yl)urea
1-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}azetidin-3-ol
5-({2-[5-(oxan-2-yl)furan-2-yl]-1H-imidazol-1-yl}methyl)-3-(propan-2-yl)-1,2-oxazole
methyl 2-({5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazol-3-yl}formamido)acetate
1-methyl-4-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)-N-methyl-1,3-thiazol-2-amine
2-{4-cyclopentanecarbonyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-9-yl}acetic acid
[(3R,4R)-1-[5-(methoxymethyl)furan-2-carbonyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N,1-dimethyl-N-{2-phenyl-1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]ethyl}-1H-pyrazole-3-carboxamide
5-fluoro-2-[4-(2-methoxyethoxy)phenyl]-N,N-dimethylpyrimidin-4-amine
1-[4-(4-fluorophenyl)benzoyl]-4-(pyridin-3-ylmethyl)-1,4-diazepan-5-one
2-chloro-N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-({[(5,6,7-trimethoxy-2-phenylquinolin-3-yl)methyl]amino}methyl)benzene-1-sulfonamide
1-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-4-hydroxypiperidine-4-carboxylic acid
1-(diphenylmethyl)-4-(1H-imidazol-2-ylmethyl)piperazine
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidine
(2R,3R,6R)-5-(5-chloropyridine-3-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)acetic acid
3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-2-ethyl-6-methyl-1-(thiophen-2-ylmethyl)-1,4-dihydropyridin-4-one
[1-(1-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}piperidine-4-carbonyl)piperidin-4-yl](phenyl)methanol
N-[(1-methylpiperidin-3-yl)methyl]-3-(2-oxopyrrolidin-1-yl)-N-(2-phenylethyl)propanamide
N-benzyl-N,1-dimethyl-5-[(2,2,2-trifluoroethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}amine
5-fluoro-2-{1-[1-(propan-2-yl)piperidine-4-carbonyl]piperidin-2-yl}-1H-1,3-benzodiazole
4-[(3-methylthiophen-2-yl)methyl]-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
2-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}-2-(3-fluoro-4-methoxyphenyl)acetic acid
N-(1,2,3,4-tetrahydronaphthalen-1-yl)-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-({7-[2-(2,3-difluorophenyl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide