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N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(ethylsulfanyl)-1,3-benzoxazol-6-yl]-1-methylurea
3-cyclopropyl-N-{[7-(3,6-dimethylpyrazin-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-1H-pyrazole-5-carboxamide
1-methyl-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,4,9-triazaspiro[5.5]undecane
1-ethyl-4-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-5-(methoxymethyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
3-({[(1,3-dimethylpyrrolidin-3-yl)methyl](methyl)amino}methyl)-N-(3-methylpyridin-2-yl)benzamide
N-[(2-fluorophenyl)methyl]-3-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propanamide
7-fluoro-3-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-3-yl)ethyl]-1-benzofuran-2-carboxamide
1-ethyl-N-[(4-methoxyphenyl)methyl]-5-(5-methylpyrazine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-methoxy-1-methyl-2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-indole
N-{[7-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methoxyphenoxy)acetamide
2-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-6-methylphenol
N-(furan-2-ylmethyl)-4-(3-propoxypiperidin-1-yl)pyridine-2-carboxamide
3-(morpholin-4-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N4-methyl-N2-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}pyrimidine-2,4-diamine
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-(4-ethylpiperazin-1-yl)-N-(pyridin-3-ylmethyl)acetamide
methyl 1-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetyl}piperidine-2-carboxylate
2-{[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-phenyl-1,3-thiazole
{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-methoxyethyl)(propan-2-yl)amine
(3S)-4-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-1-ethyl-3-methylpiperazin-2-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[2-(3-methoxypropyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-methylpiperidine-3-carboxamide
N-[2-(2-methoxyphenyl)ethyl]-2-[4-(4-{methyl[1-(1,3-thiazol-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
7-(oxan-4-yl)-2-(2-phenoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
8-(3-hydroxypropanoyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-butyl-N-methyl-N-[2-(pyridin-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
1-[1-(4-chloro-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
3-(1H-imidazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}butanamide
1-[(2-methylphenyl)methyl]-5-{2-[(prop-2-en-1-yl)amino]ethyl}pyrrolidin-2-one
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-methylphenyl)sulfanyl]piperidine
N-[2-(6-fluoro-1H-1,3-benzodiazol-2-yl)ethyl]-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-6-oxo-1,6-dihydropyridine-2-carboxamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[2-(dimethylamino)ethyl]-N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-[(3S,4R)-1-(1-acetylpiperidine-4-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide
1-[(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}thiophen-3-yl)methyl]pyrrolidine
3-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepane-1-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1H-indol-4-one
N-[(2R,3R)-2-methoxy-1'-(3-methylbenzoyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenylacetamide
6-cyclopentyl-3-{[(5-ethylpyrimidin-2-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[(2E)-3-phenylprop-2-en-1-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-[(4-methyl-1H-imidazol-5-yl)methyl]-2-(2-phenylethyl)morpholine
6-ethoxy-4-methyl-2-[4-(thian-4-yl)-1,4-diazepan-1-yl]quinazoline
8-chloro-N-[(1-methylpyrrolidin-3-yl)methyl]quinoline-2-carboxamide
N2-[2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine
4-(cyclopropylmethyl)-2-[(4-methoxyphenyl)methyl]morpholine
2-[(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-decahydroisoquinolin-2-yl]-5,6,7,8-tetrahydroquinoline
ethyl 3-[(3-methoxyphenyl)methyl]-1-(pyridin-2-ylmethyl)piperidine-3-carboxylate
2-[(3-methoxyphenyl)methyl]-8-(1,2-oxazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
dimethyl(1-{1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}ethyl)amine