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4-{1-[(5-fluoro-2-methylphenyl)methyl]-1H-imidazol-2-yl}benzene-1,2-diol
2-(3,4-dichlorophenyl)-4-(6-methoxypyrimidin-4-yl)morpholine
(1R,5R)-3-(3,4-dimethoxybenzenesulfonyl)-6-methyl-3,6-diazabicyclo[3.2.2]nonane
N-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
9-methoxy-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(methylamino)-N-[2-(pyridin-3-ylformamido)ethyl]pyridine-4-carboxamide
2-{[(5-{1-[(2-aminopyridin-3-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
(3S,4R)-1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-methylpiperidine-3,4-diol
[2-(3-chlorophenyl)ethyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1,3-dimethyl-N-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3aS,6aS)-N-methyl-5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-N-phenyl-octahydropyrrolo[2,3-c]pyrrole-1-carboxamide
2-[5-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]-1-propyl-1H-imidazole
1-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-3-(1,2,3-thiadiazol-5-yl)urea
4-methoxy-2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}phenol
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)pent-4-enamide
1-(furan-2-ylmethyl)-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}piperidine-3-carboxamide
2-butyl-8-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]acetamide
5-[4-(difluoromethoxy)phenyl]-1,2,3,4-tetrahydroisoquinoline
2-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidin-1-yl]-6-phenylpyridine-3-carboxylic acid
(3aS,6aS)-5-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1-methyl-octahydropyrrolo[3,4-b]pyrrole
N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2-(pyridin-2-ylsulfanyl)acetamide
3-methyl-1-[1-(6-{methyl[2-(methylamino)ethyl]amino}pyridine-3-carbonyl)piperidin-3-yl]butan-1-one
N-(4-fluorophenyl)-1-(7-methyl-1-benzofuran-2-carbonyl)piperidin-3-amine
(2R,3S,6R)-3-phenyl-5-(1-propyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(4-methoxyphenyl)methyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]morpholine-4-carboxamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
3-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
3-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
4-[(4-methoxyphenyl)methyl]-1-(2-methylbenzoyl)-1,4-diazepan-5-one
8-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
(3aR,5S,6S,7aS)-2-[(1-propyl-1H-pyrazol-4-yl)sulfonyl]-octahydro-1H-isoindole-5,6-diol
N-(2-fluorophenyl)-3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}propanamide
7-(2,6-dimethoxyphenyl)-9-methoxy-4-(pyridine-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(hydroxymethyl)-N-{3-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}azepane-1-carboxamide
5-(6-chloro-2H-1,3-benzodioxol-5-yl)-3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-ethyl-3-[(1-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}piperidin-4-yl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-methyl-N-(2-phenoxyethyl)azepane-2-carboxamide
N-(1-{[(3,3-diphenylpropyl)carbamoyl]methyl}-1H-pyrazol-4-yl)-3-(2-methoxyphenyl)propanamide
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
(5S,9aS,9bS)-5-(4-methoxynaphthalen-1-yl)-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(carbamoylmethyl)-N-{[2-chloro-5-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-methyl-9-(morpholine-4-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
4-benzyl-3-ethyl-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1,4-diazepan-5-one
6-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
(9aR)-2-methyl-8-(4-phenylbenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(5S,9aS,9bS)-5-(4-phenyl-1,3-thiazol-2-yl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(1-ethyl-5-{spiro[2.4]heptane-1-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl)-4-phenylpiperazine
2-{1-[4-(3-methylphenoxy)benzoyl]azetidin-3-yl}pyridine