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5-methyl-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N,N-dimethyl-4-[4-(pyridin-4-ylmethyl)-1,4-diazepane-1-carbonyl]aniline
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-4H-thieno[3,2-b]pyrrole-5-carboxamide
N-benzyl-N-[(1R,2R)-2-hydroxycyclohexyl]imidazo[1,2-a]pyridine-6-carboxamide
N-{[3-(cyclopentyloxy)-4-methoxyphenyl]methyl}-4-phenyl-N-(pyridin-4-ylmethyl)benzamide
3-[(oxolan-3-ylmethyl)sulfamoyl]-N-[2-(1H-pyrazol-1-yl)ethyl]benzamide
3-[(3S,7S,8aS)-3-[(benzyloxy)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-chlorophenyl)urea
1-({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)-4-(3-methoxypropyl)piperidine
4-methyl-2-[1-(5-methylthiophene-3-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
6-methyl-5-{5-[2-methyl-6-(2-methylpropyl)pyrimidin-4-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
N-[2-methoxy-5-({methyl[1-(pyridin-3-yl)pentyl]carbamoyl}amino)phenyl]acetamide
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)oxolane-3-carboxamide
(2E)-3-(2-chlorophenyl)-1-{4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}prop-2-en-1-one
1-(4-chloro-3-methylphenyl)-3-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]urea
N-(2-hydroxypyridin-3-yl)-4-phenylazepane-1-carboxamide
{5-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]pyridin-2-yl}methanamine
2-{1-[2-(3-fluorophenyl)-1,3-benzoxazole-5-carbonyl]piperidin-2-yl}ethan-1-ol
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-3-yl}propanamide
{1-[(5-butylthiophen-2-yl)methyl]-3-ethylpiperidin-3-yl}methanol
1-cyclobutanecarbonyl-4-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]piperidine
{4-[(4-methoxyphenyl)methyl]-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}methanol
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-bis(2-methylpropyl)acetamide
2-(2,3-dihydro-1H-inden-1-yl)-N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]acetamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(5-methylfuran-2-yl)methyl]piperidine
2-{4-[(2-methoxyethyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}pyridine-4-carboxamide
1-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-3-(1H-pyrazol-1-yl)propan-1-one
N-({5-methyl-2-[3-(3-methylbutanamido)phenyl]-1,3-oxazol-4-yl}methyl)quinoxaline-5-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-(2-oxopyrrolidin-1-yl)propanamide
5-(2,6-dimethoxyphenyl)-N-[2-(3-methoxyphenyl)ethyl]-1,2,4-triazin-3-amine
5-chloro-3-[(4-methyl-1H-imidazol-2-yl)methyl]-3,4-dihydroquinazolin-4-one
1-(2-fluorophenyl)-4-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}piperazine
dimethyl({3-[2-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]propyl})amine
N-({3-[3-(dimethylamino)propoxy]-4-methoxyphenyl}methyl)-3-methyl-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
4-({[4-(butan-2-yloxy)-3-methoxyphenyl]methyl}amino)-N-ethylpiperidine-1-carboxamide
1-cyclohexyl-4-{3-[(3,4-dimethylpiperazin-1-yl)methyl]imidazo[1,2-a]pyridine-2-carbonyl}piperazine
2-(2-{[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
3-{[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
3-chloro-6-methyl-N-{2-[2-(propan-2-yloxy)phenyl]ethyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N6-cyclopropyl-N4-methyl-N4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]pyrimidine-2,4,6-triamine
5-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridine-2-carbonitrile
N3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
1-(3-fluoro-4-methoxybenzoyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
5-(morpholin-4-ylmethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)furan-3-carboxamide
{[(3S,4R)-1-(1H-imidazol-4-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl}dimethylamine
2-[(4-methoxyphenyl)methyl]-4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}morpholine
5-{[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}-2-(propan-2-yl)pyrimidine
1-[3-fluoro-5-(trifluoromethyl)phenyl]-3-[3-(1H-1,2,3-triazol-1-yl)propyl]urea
1-(azocan-1-yl)-3-[2-methoxy-5-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-(1H-imidazol-1-yl)-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]benzamide